SCHEMBL7832793

SCHEMBL7832793

O=NC(=O)Cc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.58
CES2 O00748 1/20 0.58
AKR1B1 P15121 1/20 0.58
CTBP2 P56545 1/20 0.52
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
FNTA P49354 1/20 0.48
FNTB P49356 1/20 0.48
HIF1A Q16665 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPK1 P28482 1/20 0.47
EPHX2 P34913 1/20 0.47
PAM P19021 2/20 0.45
TSHR P16473 2/20 0.45
ABCC4 O15439 1/20 0.45
LMNA P02545 1/20 0.45
GAA P10253 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14997451 0.84 CA2 (0.58) AKR1B1MEN1KMT2AHIF1AALDH1A1
SCHEMBL699924 0.83 CES1 (0.61) CES1CES2AKR1B1CTBP2MEN1
SCHEMBL1300068 0.79 CES1 (0.56) CES1CES2AKR1B1CTBP2MEN1
SCHEMBL15241380 0.79 CES1 (0.56) CES1CES2AKR1B1CTBP2MEN1
SCHEMBL15372403 0.77 CES2 (0.44) CES1CES2AKR1B1CTBP2FNTA
SCHEMBL7431387 0.77 CYP19A1 (0.46) ALDH1A1GAAHTTMAPTMET
SCHEMBL16519727 0.77 KEAP1 (0.61) KMT2AHDAC8HDAC6ALDH1A1MAPK1
SCHEMBL8013340 0.77 CES1 (0.54) CES1CES2AKR1B1CTBP2MEN1
SCHEMBL13017398 0.77 CTBP2 (0.53) CTBP2MEN1KMT2AHDAC8HDAC6
SCHEMBL17040103 0.77 GFER (0.42) ALDH1A1TSHRCYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9988665-B2 Methods for determining protein binding specificity using peptide libraries WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2018-06-05 US disclosed
EP-2328865-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-05-31 EP disclosed
CN-103596929-B Pyrazole and pyrimidine tricycloalkenones as antioxidant inflammation modulators 里亚塔医药公司 2016-10-19 CN disclosed
US-20160115145-A1 ROSEOBACTICIDES AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2016-04-28 US disclosed
WO-2015071493-A1 CHEMOENZYMATIC SYNTHESIS OF THE CEPHALOSPORINE INTERMEDIATE 7-AMINO-3-ALKENYLCEPHEM-4-CARBOXYLIC ACID SANDOZ AG (CH) 2015-05-21 WO disclosed
WO-2013163466-A1 INHIBITORS OF HEPATITIS C VIRUS PRESIDIO PHARMACEUTICALS, INC. (US) 2013-10-31 WO disclosed
WO-2010055136-A1 PROCESS FOR THE PURIFICATION OF ANTIBODIES USING AFFINITY RESINS COMPRISING SPECIFIC LIGANDS NOVO NORDISK A/S (DK) 2010-05-20 WO disclosed
EP-1091938-A2 ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF Aventis Pharmaceuticals Inc. (US) 2001-04-18 EP disclosed
WO-2000001671-A2 ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF AVENTIS PHARMACEUTICALS INC. (US) 2000-01-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160115145-A1 ROSEOBACTICIDES AND USES THEREOF CROCC, MRPL21, RPL41 CES1 4119/4885CES2 420/4885AKR1B1 3679/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.