SCHEMBL7833632

SCHEMBL7833632

CC(C)(C)OC(=O)Nn1c(C(=O)O)cc2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.50
DAO P14920 1/20 0.48
ALDH1A1 P00352 3/20 0.46
TSHR P16473 1/20 0.46
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CCR2 P41597 3/20 0.43
NR1H2 P55055 8/20 0.42
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
KDM4A O75164 1/20 0.40
NR1H3 Q13133 2/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
GAA P10253 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551062 0.87 MCL1 (0.57) MCL1DAOALDH1A1TSHRKDM4E
SCHEMBL27896993 0.83 SLC9A1 (0.39) MCL1MEN1NPC1GAARAB9A
SCHEMBL10379817 0.79 DAO (0.59) MCL1DAOALDH1A1TSHRKDM4E
SCHEMBL9120939 0.77 CCR2 (0.51) MCL1DAOALDH1A1TSHRCCR2
SCHEMBL29781083 0.76 NR1H2 (0.55) MCL1DAOALDH1A1TSHRNR1H2
SCHEMBL7902953 0.76 NR1H2 (0.55) MCL1DAOALDH1A1TSHRNR1H2
SCHEMBL25195634 0.75 MCL1 (0.53) MCL1DAOALDH1A1TSHRKDM4E
SCHEMBL5728166 0.73 MCL1 (0.50) MCL1DAOALDH1A1TSHRKDM4E
SCHEMBL3958982 0.73 CCR2 (0.56) MCL1DAOALDH1A1TSHRKDM4E
SCHEMBL4098402 0.73 CTSS (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0918752-A4 DNA-BINDING INDOLE DERIVATIVES, THEIR PRODRUGS AND IMMUNOCONJUGATES AS ANTICANCER AGENTS PANORAMA RES INC (US) 2001-11-21 EP disclosed
EP-0918752-A2 DNA-BINDING INDOLE DERIVATIVES, THEIR PRODRUGS AND IMMUNOCONJUGATES AS ANTICANCER AGENTS PANORAMA RESEARCH, INC. (US) 1999-06-02 EP disclosed
WO-1997044000-A2 DNA-BINDING INDOLE DERIVATIVES, THEIR PRODRUGS AND IMMUNOCONJUGATES AS ANTICANCER AGENTS PANORAMA RESEARCH, INC. (US) 1997-11-27 WO disclosed