SCHEMBL7833683

SCHEMBL7833683

COc1ccccc1N1CCN(CCCn2cc(C)c(=O)[nH]c2=O)CC1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 2/20 0.75
ADRA1A P35348 2/20 0.75
ADRA1B P35368 2/20 0.75
DRD2 P14416 3/20 0.62
DRD3 P35462 3/20 0.62
HTR7 P34969 7/20 0.61
HTR1A P08908 5/20 0.61
ALDH1A1 P00352 2/20 0.59
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2D6 P10635 1/20 0.59
ALOX12 P18054 1/20 0.59
HIF1A Q16665 1/20 0.59
HSD17B10 Q99714 1/20 0.59
KDM4E B2RXH2 1/20 0.58
GLA P06280 1/20 0.58
HPGD P15428 1/20 0.58
CYP1A2 P05177 1/20 0.57
CYP2C9 P11712 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7834507 0.99 ADRA1D (0.74) ADRA1DADRA1AADRA1BDRD2DRD3
SCHEMBL2350823 0.98 ADRA1D (0.72) ADRA1DADRA1AADRA1BDRD2DRD3
SCHEMBL2351486 0.87 ADRA1B (0.75) ADRA1DADRA1AADRA1BDRD2HTR7
Hydrochloric Acid SCHEMBL7833133 0.87 ADRA1A (0.64) ADRA1DADRA1AADRA1BDRD2DRD3
SCHEMBL2353857 0.86 ADRA1B (0.68) ADRA1DADRA1AADRA1BDRD2DRD3
Hydrochloric Acid SCHEMBL7831192 0.85 ADRA1D (0.59) ADRA1DADRA1AADRA1BDRD2DRD3
Hydrochloric Acid SCHEMBL9045935 0.85 ADRA1A (0.98) ADRA1DADRA1AADRA1BDRD2DRD3
SCHEMBL2354965 0.84 ADRA1A (0.66) ADRA1DADRA1AADRA1BDRD2DRD3
SCHEMBL2349477 0.84 ADRA1D (0.58) ADRA1DADRA1AADRA1BDRD2DRD3
SCHEMBL2351537 0.84 ADRA1B (0.55) ADRA1DADRA1AADRA1BDRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748800-B1 Pyrimidinedione, pyrimidinetrione, triazinedione derivatives as alpha-1-adrenergic receptor antagonists HOFFMANN LA ROCHE (CH) 2001-05-09 EP disclosed
EP-0748800-A2 Pyrimidinedione, pyrimidinetrione, triazinedione, tetrahydroquinazolinedione derivatives as alpha-1-adrenergic receptor antagonists F. HOFFMANN-LA ROCHE AG (CH) 1996-12-18 EP disclosed