SCHEMBL7833964

SCHEMBL7833964

CCCc1cn(Cc2ccccc2)c(=O)n(CCCN2CCN(c3ccccc3OC)CC2)c1=O

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.53
DRD3 P35462 3/20 0.53
HTR1A P08908 2/20 0.53
ADRA1D P25100 2/20 0.53
ADRA1A P35348 1/20 0.53
ADRA1B P35368 1/20 0.53
HTR7 P34969 2/20 0.52
SLC6A2 P23975 1/20 0.51
SLC6A4 P31645 1/20 0.51
ADRB2 P07550 1/20 0.50
ADRA2A P08913 1/20 0.50
ADRA2B P18089 1/20 0.50
ADRA2C P18825 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7835944 0.99 DRD2 (0.53) DRD2DRD3HTR1AADRA1DADRA1A
SCHEMBL7822356 0.94 DRD2 (0.55) DRD2DRD3HTR1AADRA1DADRA1A
Hydrochloric Acid SCHEMBL7821312 0.93 DRD2 (0.54) DRD2DRD3HTR1AADRA1DADRA1A
SCHEMBL7833750 0.91 HTR7 (0.56) DRD2DRD3HTR1AADRA1DADRA1A
SCHEMBL7830170 0.88 ADRA1A (0.57) DRD2DRD3ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL7821711 0.88 ADRA1A (0.57) DRD2DRD3ADRA1DADRA1AADRA1B
SCHEMBL7830329 0.87 HTR1A (0.56) DRD2DRD3HTR1AADRA1DADRA1A
Hydrochloric Acid SCHEMBL7821236 0.86 HTR1A (0.55) DRD2DRD3HTR1AADRA1DADRA1A
SCHEMBL7821704 0.84 HTR7 (0.52) DRD2DRD3HTR1AADRA1DADRA1A
Hydrochloric Acid SCHEMBL7830388 0.83 HTR7 (0.52) DRD2DRD3HTR1AADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748800-B1 Pyrimidinedione, pyrimidinetrione, triazinedione derivatives as alpha-1-adrenergic receptor antagonists HOFFMANN LA ROCHE (CH) 2001-05-09 EP disclosed
US-5859014-A USEFUL IN TREATMENT OF DISEASES INVOLVING DIRECTLY OR INDIRECTLY AN OBSTRUCTION OF THE LOWER URINARY TRACT, SUCH ASBENIGN PROSTATE HYPERPLASIA SYNTEX (U.S.A.) INC. (US) 1999-01-12 US disclosed
EP-0748800-A2 Pyrimidinedione, pyrimidinetrione, triazinedione, tetrahydroquinazolinedione derivatives as alpha-1-adrenergic receptor antagonists F. HOFFMANN-LA ROCHE AG (CH) 1996-12-18 EP disclosed