SCHEMBL7834261

SCHEMBL7834261

CSc1ccc2[nH]c(CCCCl)c(C=O)c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
MAPT P10636 2/20 0.46
HPGD P15428 2/20 0.46
GAA P10253 1/20 0.46
TSHR P16473 1/20 0.46
HSD17B10 Q99714 1/20 0.46
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
RAB9A P51151 1/20 0.36
HTR6 P50406 3/20 0.35
HTR3E A5X5Y0 2/20 0.35
HTR3B O95264 2/20 0.35
HTR1A P08908 2/20 0.35
HTR1D P28221 2/20 0.35
HTR1B P28222 2/20 0.35
HTR2A P28223 2/20 0.35
HTR2C P28335 2/20 0.35
HTR1E P28566 2/20 0.35
HTR1F P30939 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7835267 0.87 ALDH1A1 (0.46) ALDH1A1KDM4EMAPTHPGDGAA
SCHEMBL7835119 0.83 MAPT (0.42) ALDH1A1KDM4EMAPTHPGDGAA
SCHEMBL7834309 0.81 AHR (0.51) ALDH1A1MAPTHPGDGAALMNA
SCHEMBL7835647 0.80 AHR (0.53) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL7836059 0.76 AHR (0.54) ALDH1A1MAPTHSD17B10LMNAPOLB
SCHEMBL7837899 0.76 AHR (0.52) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL7834834 0.75 AHR (0.51) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL7836031 0.74 PDE7A (0.36) AHR
SCHEMBL7836341 0.72 MAOA (0.53) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL7835639 0.70 ALDH1A1 (0.36) ALDH1A1KDM4EHPGDGAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109813-A1 PYRROLOINDOLES, PYRIDOINDOLES AND AZEPINOINDOLES AS 5-HT2C AGONISTS VERNALIS RESEARCH LIMITED (GB) 2001-06-27 EP disclosed
WO-2000012510-A1 PYRROLOINDOLES, PYRIDOINDOLES AND AZEPINOINDOLES AS 5-HT2C AGONISTS VERNALIS RESEARCH LIMITED (GB) 2000-03-09 WO disclosed