SCHEMBL7836059

SCHEMBL7836059

O=Cc1c(CCCCl)[nH]c2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AHR P35869 6/20 0.54
KMT2A Q03164 2/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
KIF11 P52732 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MITF O75030 1/20 0.38
LMNA P02545 1/20 0.38
RAB9A P51151 1/20 0.38
POLB P06746 1/20 0.38
CYP2A6 P11509 1/20 0.38
GSK3B P49841 2/20 0.36
HKDC1 Q2TB90 1/20 0.36
GPR3 P46089 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7834309 0.81 AHR (0.51) AHRKMT2AMAPTMEN1ALDH1A1
SCHEMBL9395996 0.81 AHR (0.50) AHRALDH1A1HSD17B10
SCHEMBL1536184 0.81 AHR (0.50) AHRKMT2AMAPTMEN1ALDH1A1
SCHEMBL7835119 0.80 MAPT (0.42) AHRKMT2AMAPTMEN1ALDH1A1
SCHEMBL7834282 0.78 AHR (0.41) AHRKMT2AMEN1ALDH1A1
SCHEMBL7836341 0.77 MAOA (0.53) KMT2AMAPTMEN1ALDH1A1RAB9A
SCHEMBL14199367 0.77 AHR (0.43) AHRKMT2AMAPTMEN1KIF11
SCHEMBL7493848 0.77 AHR (0.52) AHRKMT2AMAPTMEN1KIF11
SCHEMBL29951745 0.77 AHR (0.59) AHRKMT2AMAPTMEN1KIF11
SCHEMBL9274962 0.77 AHR (0.59) AHRKMT2AMAPTMEN1KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109813-A1 PYRROLOINDOLES, PYRIDOINDOLES AND AZEPINOINDOLES AS 5-HT2C AGONISTS VERNALIS RESEARCH LIMITED (GB) 2001-06-27 EP disclosed
WO-2000012510-A1 PYRROLOINDOLES, PYRIDOINDOLES AND AZEPINOINDOLES AS 5-HT2C AGONISTS VERNALIS RESEARCH LIMITED (GB) 2000-03-09 WO disclosed