SCHEMBL7834309

SCHEMBL7834309

O=Cc1c(CCCCl)[nH]c2ccc(Cl)cc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 2/20 0.51
LMNA P02545 1/20 0.42
SIRT1 Q96EB6 8/20 0.41
SIRT2 Q8IXJ6 1/20 0.39
CYP1A2 P05177 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.37
UTS2R Q9UKP6 1/20 0.36
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
HTR7 P34969 1/20 0.36
HTR2B P41595 1/20 0.36
HTR6 P50406 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7835119 0.84 MAPT (0.42) AHRLMNAGAAHPGDALOX15
SCHEMBL7835647 0.81 AHR (0.53) AHRLMNACYP1A2HPGDHTR7
SCHEMBL7834261 0.81 ALDH1A1 (0.46) AHRLMNAGAAHPGDHTR7
SCHEMBL7836059 0.81 AHR (0.54) AHRLMNAMEN1ALDH1A1MAPT
SCHEMBL7836031 0.78 PDE7A (0.36) AHRMPOXDH
SCHEMBL7837899 0.78 AHR (0.52) AHRLMNACYP1A2HPGDHTR7
SCHEMBL7834834 0.77 AHR (0.51) AHRLMNACYP1A2HPGDHTR7
SCHEMBL7836341 0.76 MAOA (0.53) CYP1A2HPGDMEN1ALDH1A1MAPT
SCHEMBL22898794 0.75 LMNA (0.51) AHRLMNACYP1A2GAAHPGD
SCHEMBL29363428 0.75 LMNA (0.51) AHRLMNACYP1A2GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109813-A1 PYRROLOINDOLES, PYRIDOINDOLES AND AZEPINOINDOLES AS 5-HT2C AGONISTS VERNALIS RESEARCH LIMITED (GB) 2001-06-27 EP disclosed
WO-2000012510-A1 PYRROLOINDOLES, PYRIDOINDOLES AND AZEPINOINDOLES AS 5-HT2C AGONISTS VERNALIS RESEARCH LIMITED (GB) 2000-03-09 WO disclosed