SCHEMBL7834503

SCHEMBL7834503

N#CCc1nc2cc(-n3ccnc3)ccc2[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.43
CYP11B1 P15538 2/20 0.43
CYP11B2 P19099 2/20 0.43
F9 P00740 1/20 0.43
CBFB Q13951 1/20 0.42
NCOA3 Q9Y6Q9 1/20 0.42
FGFR1 P11362 1/20 0.39
FLT1 P17948 1/20 0.39
PGR P06401 1/20 0.39
PDE2A O00408 1/20 0.38
PDE1A P54750 1/20 0.38
PDE1B Q01064 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE1C Q14123 1/20 0.38
PDE3A Q14432 1/20 0.38
MAOA P21397 3/20 0.38
MAOB P27338 3/20 0.38
IDH1 O75874 1/20 0.38
KCNMA1 Q12791 1/20 0.38
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7834506 0.90 CBFB (0.53) CYP19A1CYP11B1CYP11B2F9CBFB
Hydrochloric Acid SCHEMBL8155236 0.82 F9 (0.46) CYP19A1CYP11B1CYP11B2F9CBFB
SCHEMBL7407358 0.80 CBFB (0.50) CYP19A1CYP11B1CYP11B2F9CBFB
SCHEMBL7834248 0.79 F9 (0.46) CYP19A1CYP11B1CYP11B2F9CBFB
SCHEMBL7821986 0.76 NPC1 (0.55) CYP19A1CYP11B1CYP11B2F9CBFB
SCHEMBL7821729 0.76 RAB9A (0.55) CYP19A1CYP11B1CYP11B2CBFBNCOA3
SCHEMBL7822768 0.76 IDH1 (0.48) CYP19A1CYP11B1CYP11B2F9CBFB
SCHEMBL7832698 0.76 F9 (0.42) CYP19A1CYP11B1CYP11B2F9CBFB
SCHEMBL14162135 0.76 FGFR1 (0.49) CYP19A1CYP11B1CYP11B2F9CBFB
SCHEMBL7833749 0.75 MEN1 (0.46) CYP19A1CYP11B1CYP11B2F9CBFB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894795-B1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-06 EP disclosed
US-6040327-A INHIBITORS OF INTERLEUKINS; TREATING RHEUMATOID ARTHRITIS OR ARTHROSIS ADIR ET COMPAGNIE (FR) 2000-03-21 US disclosed
EP-0894795-A1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-02-03 EP disclosed