SCHEMBL7835692

SCHEMBL7835692

CCNc1cc(F)cc(C(F)(F)F)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 6/20 0.51
EGFR P00533 3/20 0.42
PTPN5 P54829 1/20 0.41
CYP1A2 P05177 2/20 0.40
S1PR2 O95136 1/20 0.40
SMYD2 Q9NRG4 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
IDH1 O75874 1/20 0.39
PPARA Q07869 1/20 0.38
MAPT P10636 1/20 0.37
RAPGEF4 Q8WZA2 1/20 0.37
GRM4 Q14833 1/20 0.37
P2RX1 P51575 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27668287 0.98 TRPA1 (0.50) TRPA1EGFRPTPN5CYP1A2S1PR2
SCHEMBL4966922 0.88 TRPA1 (0.53) TRPA1PTPN5CYP1A2MAPTRAPGEF4
SCHEMBL7868346 0.85 TRPA1 (0.47) TRPA1EGFRPTPN5CYP1A2IDH1
SCHEMBL3959091 0.81 RAPGEF4 (0.40) TRPA1CYP1A2PPARAMAPTRAPGEF4
SCHEMBL10104509 0.81 RAPGEF4 (0.49) TRPA1PTPN5CYP1A2MAPTRAPGEF4
SCHEMBL22312230 0.79 RAPGEF4 (0.53) TRPA1PTPN5CYP1A2HDAC3HDAC1
SCHEMBL21571898 0.78 EGFR (0.40) TRPA1EGFRS1PR2HDAC3HDAC1
SCHEMBL7944387 0.78 KIF11 (0.45) EGFRS1PR2HDAC3HDAC1HDAC2
SCHEMBL21571897 0.77 EGFR (0.40) TRPA1EGFRCYP1A2S1PR2SMYD2
SCHEMBL8168077 0.77 DHFR (0.46) TRPA1PTPN5HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1165531-C Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing phenylenediamine groups 2004-09-08 CN disclosed
CN-1367785-A Heterocyclic carboxamide-containing thiourea inhibitors of herpes viruses containing substituted phenylenediamine groups AMERICAN HOME PROD (US) 2002-09-04 CN disclosed
CN-1348446-A Heterocyclic carboxamide-containing thiourea inhibitors of herpes viruses containing phenylenediamine groups AMERICAN HOME PROD (US) 2002-05-08 CN disclosed
CN-1335843-A Thiourea inhibitors of herpes viruses AMERICAN HOME PROD (US) 2002-02-13 CN disclosed
CN-1333769-A Thiourea inhibitors of herps viruses AMERICAN HOME PROD (US) 2002-01-30 CN disclosed
CN-1333750-A Acetamide and substituted acetamide-containing thiourea inhibitors of herpes viruses AMERICAN HOME PROD (US) 2002-01-30 CN disclosed
CN-1329608-A Alpha-methylbenzyl-containing thioure a inhibitors of herpes viruses containing phenylenediamine group AMERICAN HOME PROD (US) 2002-01-02 CN disclosed
EP-1137647-A1 THIOUREA INHIBITORS OF HERPES VIRUSES AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-04 EP disclosed
WO-2000034268-A1 THIOUREA INHIBITORS OF HERPES VIRUSES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed