SCHEMBL7836697

SCHEMBL7836697

CCCCC(CO)(CCCC)NS(=O)(=O)c1ccc(N(C)C)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
TDP1 Q9NUW8 2/20 0.43
MAPT P10636 2/20 0.43
MAPK1 P28482 2/20 0.43
MCL1 Q07820 2/20 0.43
LMNA P02545 1/20 0.43
GFER P55789 1/20 0.43
KEAP1 Q14145 1/20 0.43
NFE2L2 Q16236 1/20 0.43
CA9 Q16790 1/20 0.42
FLT1 P17948 2/20 0.42
FLT4 P35916 2/20 0.42
KDR P35968 2/20 0.42
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC11 Q96DB2 1/20 0.39
F2 P00734 1/20 0.39
PRSS1 P07477 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7838172 0.83 FFAR1 (0.50) ALDH1A1MAPK1LMNAHDAC3HDAC1
SCHEMBL7846693 0.75 LIMK1 (0.33) ALDH1A1MAPTMAPK1MCL1LMNA
SCHEMBL7837233 0.72 MEN1 (0.35) ALDH1A1MAPTMAPK1LMNAGFER
SCHEMBL25754608 0.71 ALDH1A1 (0.56) ALDH1A1TDP1MAPTMAPK1MCL1
SCHEMBL6014530 0.70 HTR6 (0.49) ALDH1A1MAPTLMNARAB9AKDM4E
SCHEMBL12284487 0.70 ALDH1A1 (0.56) ALDH1A1MAPTLMNACA9RAB9A
SCHEMBL12169312 0.69 ALDH1A1 (0.51) ALDH1A1MAPTLMNACA9HPGD
SCHEMBL11859735 0.69 CYP2C9 (0.72) ALDH1A1TDP1LMNAFLT1FLT4
SCHEMBL12509428 0.68 UCHL1 (0.51) ALDH1A1MAPTLMNAHPGDSMN1; SMN2
SCHEMBL19563499 0.68 CA1 (0.49) ALDH1A1MAPK1F2PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1155007-A2 1,2-BENZOTHIAZEPINES FOR THE TREATMENT OF HYPERLIPIDEMIC DISEASES G.D. Searle LLC (US) 2001-11-21 EP disclosed
WO-2000047568-A2 1,2-BENZOTHIAZEPINES FOR THE TREATMENT OF HYPERLIPIDEMIC DISEASES G.D. SEARLE LLC (US) 2000-08-17 WO disclosed