Oxindole

Oxindole

SCHEMBL7836705

CC1(C)C=Nc2ccccc21.O=C1Cc2ccccc2N1

nearest known ligand 0.58

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 3/20 0.58
PDK2 Q15119 1/20 0.58
NPC1 O15118 3/20 0.41
MAPK13 O15264 1/20 0.41
MAPK12 P53778 1/20 0.41
MAPK11 Q15759 1/20 0.41
MAPK14 Q16539 1/20 0.41
ALDH1A1 P00352 2/20 0.40
BRD4 O60885 1/20 0.40
CREBBP Q92793 1/20 0.40
MAPT P10636 4/20 0.40
SRC P12931 2/20 0.39
CMA1 P23946 2/20 0.39
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
GRIA1 P42261 2/20 0.38
CACNG8 Q8WXS5 2/20 0.38
EIF2AK2 P19525 1/20 0.38
CASP3 P42574 2/20 0.37
MEN1 O00255 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxindole SCHEMBL1144643 0.76 AHR (1.00) AHRPDK2NPC1MAPK13MAPK12
SCHEMBL926937 0.76 HTR5A (0.35) PDK2CASP3RAB9ASENP8SENP7
SCHEMBL29639106 0.76 HTR5A (0.35) PDK2CASP3RAB9ASENP8SENP7
Oxindole SCHEMBL29358826 0.76 AHR (1.00) AHRPDK2NPC1MAPK13MAPK12
Oxindole SCHEMBL19504 0.76 AHR (1.00) AHRPDK2NPC1MAPK13MAPK12
Oxindole SCHEMBL15636313 0.75 AHR (0.95) AHRPDK2NPC1MAPK13MAPK12
Oxindole SCHEMBL5502064 0.75 AHR (0.95) AHRPDK2NPC1MAPK13MAPK12
Oxindole SCHEMBL4720301 0.75 AHR (0.95) AHRPDK2NPC1MAPK13MAPK12
Oxindole SCHEMBL5624006 0.75 AHR (0.95) AHRPDK2NPC1MAPK13MAPK12
Oxindole SCHEMBL1462135 0.75 AHR (0.95) AHRPDK2NPC1MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780388-B1 5HT1Dalpha and 5HT2A ligands LILLY CO ELI (GB) 2001-08-16 EP disclosed
US-5773448-A NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY LIMITED (GB) 1998-06-30 US disclosed
EP-0780388-A1 5HT1Dalpha and 5HT2A ligands LILLY INDUSTRIES LIMITED (GB) 1997-06-25 EP disclosed