SCHEMBL7836741

SCHEMBL7836741

CC(C)(C(=O)O)C(NC(=O)c1ccc(C#N)cc1)c1cccc(Cl)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 4/20 0.62
CTSG P08311 4/20 0.62
CTRB1 P17538 4/20 0.62
CMA1 P23946 4/20 0.62
ITGB3 P05106 2/20 0.48
ITGA2B P08514 2/20 0.48
CNR1 P21554 2/20 0.47
CNR2 P34972 2/20 0.47
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
SLC6A9 P48067 1/20 0.46
SLC6A5 Q9Y345 1/20 0.46
CTSV O60911 2/20 0.44
CTSL P07711 2/20 0.44
CTSB P07858 2/20 0.44
CTSS P25774 2/20 0.44
CTSK P43235 2/20 0.44
TRPA1 O75762 3/20 0.43
S1PR3 Q99500 4/20 0.43
S1PR4 O95977 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7825862 0.87 CTSG (0.80) PRSS1CTSGCTRB1CMA1CYP2D6
SCHEMBL7826107 0.82 PRSS1 (0.62) PRSS1CTSGCTRB1CMA1ITGB3
SCHEMBL7836801 0.79 CTSG (0.64) PRSS1CTSGCTRB1CMA1TRPA1
SCHEMBL7837287 0.79 PRSS1 (0.64) PRSS1CTSGCTRB1CMA1CYP2C9
SCHEMBL7836737 0.78 PRSS1 (0.48) PRSS1CTSGCTRB1CMA1CNR1
SCHEMBL7836199 0.77 CTSG (0.65) PRSS1CTSGCTRB1CMA1S1PR3
SCHEMBL7835567 0.77 CTSG (0.58) PRSS1CTSGCTRB1CMA1TRPA1
SCHEMBL7835767 0.77 PRSS1 (0.56) PRSS1CTSGCTRB1CMA1TRPA1
SCHEMBL5947886 0.74 EPHX2 (0.63) CNR1CYP2D6CYP2C9SLC6A9SLC6A5
SCHEMBL7837407 0.72 PRSS1 (0.54) PRSS1CTSGCTRB1CMA1TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800516-B1 FIBRINOGEN RECEPTOR ANTAGONISTS HAVING SUBSTITUTED (b)-AMINO ACID RESIDUES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME NIPPON STEEL CORP (JP) 2001-09-19 EP disclosed
US-5866592-A Fibrinogen receptor antagonist and pharmaceutical compositions comprising the same NIPPON STEEL CORPORATION (JP) 1999-02-02 US disclosed