SCHEMBL7837255

SCHEMBL7837255

COC(=O)c1cc2ccccc2n1CC#N

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.58
MTNR1B P49286 1/20 0.58
KMT2A Q03164 2/20 0.54
NOD2 Q9HC29 1/20 0.47
NOD1 Q9Y239 1/20 0.47
MEN1 O00255 1/20 0.47
CNR2 P34972 2/20 0.46
KDM4E B2RXH2 2/20 0.45
CRHBP P24387 1/20 0.45
CRHR2 Q13324 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CCR2 P41597 1/20 0.43
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
CYP1A2 P05177 1/20 0.42
F10 P00742 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1392918 0.86 NOD2 (0.64) MTNR1AMTNR1BKMT2ANOD2NOD1
SCHEMBL7880746 0.86 MTNR1A (0.62) MTNR1AMTNR1BKMT2ANOD2NOD1
SCHEMBL30585515 0.86 NOD2 (0.64) MTNR1AMTNR1BKMT2ANOD2NOD1
SCHEMBL7425163 0.86 MTNR1A (0.58) MTNR1AMTNR1BKMT2ANOD2NOD1
SCHEMBL24170706 0.84 CCR2 (0.47) MTNR1AMTNR1BKMT2ANOD2NOD1
SCHEMBL5622129 0.84 MAPT (0.46) MTNR1AMTNR1BMAPT
SCHEMBL5622754 0.83 MTNR1A (0.61) MTNR1AMTNR1BKDM4ESMN1; SMN2CCR2
SCHEMBL29262518 0.83 F10 (0.44) MTNR1AMTNR1BKMT2AKDM4ESMN1; SMN2
SCHEMBL19252931 0.83 PTGS2 (0.45) MTNR1AMTNR1BKMT2AMAPT
SCHEMBL5917423 0.83 PTGS2 (0.46) MTNR1AMTNR1BKMT2AMEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147110-A1 PYRAZINO(AZA)INDOLE DERIVATIVES VERNALIS RESEARCH LIMITED (GB) 2001-10-24 EP disclosed
WO-2000044753-A1 PIRAZINO(AZA)INDOLE DERIVATIVES VERNALIS RESEARCH LIMITED (GB) 2000-08-03 WO disclosed