SCHEMBL7837542

SCHEMBL7837542

CC(C)C[C@@H](C(=O)NN1C(=O)NC2(CCCCC2)C1=O)[C@H](CCCc1ccccc1)C(=O)NOC1CCCCO1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 2/20 0.36
MMP13 P45452 1/20 0.36
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
MMP3 P08254 3/20 0.34
APP P05067 2/20 0.34
DGAT1 O75907 1/20 0.33
FKBP1A P62942 1/20 0.33
KMT2A Q03164 1/20 0.33
MMP2 P08253 3/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7848793 0.94 MMP1 (0.35) MMP1MMP13MMP3APPDGAT1
SCHEMBL7946535 0.93 MMP1 (0.37) MMP1MMP13L3MBTL1MMP3APP
SCHEMBL7856205 0.91 ALDH1A1 (0.38) MMP1MMP13ALDH1A1LMNAAPP
SCHEMBL7955660 0.90 XIAP (0.35) MMP1MMP13ALDH1A1LMNASMN1; SMN2
SCHEMBL6221034 0.86 MMP1 (0.38) MMP1MMP13MMP3APPFKBP1A
SCHEMBL7837114 0.86 ADAM17 (0.37) ALDH1A1LMNASMN1; SMN2L3MBTL1KMT2A
SCHEMBL7837117 0.86 ADAM17 (0.37) ALDH1A1LMNASMN1; SMN2L3MBTL1KMT2A
SCHEMBL7960600 0.84 MMP1 (0.37) MMP1MMP13MMP3APPMMP2
SCHEMBL7955118 0.84 MMP1 (0.37) MMP1MMP13MMP3APPFKBP1A
SCHEMBL7842288 0.83 MMP1 (0.37) MMP1MMP13MMP3APPMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1137640-A1 CYCLIC HYDRAZINE DERIVATIVES AS TNF-ALPHA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2001-10-04 EP disclosed
US-6281363-B1 ANTIINFLAMMATORY AGENTS; ANTIARTHRITIC AGENTS; AUTOIMMUNE DISORDERS HOFFMANN-LA ROCHE INC. 2001-08-28 US disclosed
WO-2000035885-A1 CYCLIC HYDRAZINE DERIVATIVES AS TNF-ALPHA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-22 WO disclosed