SCHEMBL7837557

SCHEMBL7837557

COc1ccc2c(c1OC)N(Cc1ccccc1Cl)C(=O)C(NC(=O)OC(C)(C)C)C2

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
XIAP P98170 6/20 0.40
TP53 P04637 2/20 0.39
MAPT P10636 1/20 0.39
CXCR6 O00574 1/20 0.39
KMT2A Q03164 4/20 0.38
MEN1 O00255 2/20 0.38
ALPL P05186 1/20 0.38
ALPI P09923 1/20 0.38
ALPG P10696 1/20 0.38
POLB P06746 1/20 0.36
THRB P10828 1/20 0.36
CCKBR P32239 1/20 0.36
NPY1R P25929 1/20 0.36
PTGER3 P43115 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7837553 0.84 XIAP (0.45) XIAPCCKBRNPY1R
SCHEMBL7848691 0.80 XIAP (0.46) XIAPCCKBRNPY1R
SCHEMBL7836160 0.79 AADAT (0.46) TP53MAPTKMT2AMEN1ALPL
SCHEMBL2847250 0.71 NPY1R (0.49) XIAPKMT2ANPY1RL3MBTL1
SCHEMBL7835962 0.70 GAA (0.43) POLB
SCHEMBL7417336 0.69 NPY1R (0.51) XIAPCCKBRNPY1RL3MBTL1
SCHEMBL2840169 0.69 NPY1R (0.47) XIAPKMT2ACCKBRNPY1RL3MBTL1
SCHEMBL5132571 0.69 NPY1R (0.59) XIAPKMT2ACCKBRNPY1RL3MBTL1
SCHEMBL7416762 0.69 NPY1R (0.59) XIAPKMT2ACCKBRNPY1RL3MBTL1
SCHEMBL7421160 0.68 SCN9A (0.48) CCKBRNPY1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802922-B1 NOVEL AMINO ACID DERIVATIVES, METHOD OF PRODUCING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM PHARMA (DE) 2001-09-26 EP disclosed
EP-0802922-A1 NOVEL AMINO ACID DERIVATIVES, METHOD OF PRODUCING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM KG (DE) 1997-10-29 EP disclosed
WO-1995023810-A1 NOVEL AMINO ACID DERIVATIVES, METHOD OF PRODUCING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM KG (DE) 1995-09-08 WO disclosed