SCHEMBL7838595

SCHEMBL7838595

N#CC(c1ccc(Cl)c(Cl)c1)c1c(Cl)cc(N)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.45
TSHR P16473 1/20 0.45
SLC6A3 Q01959 5/20 0.44
MEN1 O00255 1/20 0.36
NR1I2 O75469 1/20 0.36
KMT2A Q03164 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
IDO2 Q6ZQW0 1/20 0.36
ALDH1A1 P00352 2/20 0.34
AHR P35869 1/20 0.34
CYP2D6 P10635 3/20 0.34
SLC6A2 P23975 3/20 0.34
SLC6A4 P31645 3/20 0.34
KCNH2 Q12809 2/20 0.34
MAPT P10636 1/20 0.33
PTGS1 P23219 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8145600 0.84 MEN1 (0.48) CYP3A4SLC6A3MEN1NR1I2KMT2A
SCHEMBL7837943 0.82 SLC6A3 (0.41) CYP3A4SLC6A3MEN1NR1I2KMT2A
SCHEMBL5566385 0.82 HTT (0.39) MEN1KMT2AIDO1ALDH1A1KCNH2
SCHEMBL10672256 0.81 ALDH1A1 (0.46) CYP3A4MEN1NR1I2KMT2AIDO1
SCHEMBL7840238 0.76 HSD17B10 (0.53) CYP3A4SLC6A3MEN1NR1I2KMT2A
SCHEMBL10420876 0.74 ALDH1A1 (0.41) CYP3A4SLC6A3MEN1NR1I2KMT2A
SCHEMBL9455530 0.74 ALDH1A1 (0.45) TSHRMEN1NR1I2KMT2AALDH1A1
SCHEMBL9455449 0.73 CYP19A1 (0.41) SLC6A3MEN1NR1I2KMT2ASLC6A2
SCHEMBL11758026 0.72 CYP3A4 (0.39) CYP3A4TSHRSLC6A3MEN1KMT2A
SCHEMBL10420892 0.72 ALDH1A1 (0.43) CYP3A4MEN1NR1I2KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0737672-B1 Method of producing triazine derivatives TAKEDA SCHERING PLOUGH ANIMAL (JP) 2001-10-04 EP disclosed
US-6211178-B1 ANTIPROTOZOA AGENTS FOR COCCIDIOIDES; CYCLIZATION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US disclosed
US-5994355-A ANTIPROTOZOA AGENTS, PARASITICIDE; VETERINARY MEDICINE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-11-30 US disclosed
EP-0737672-A2 Method of producing triazine derivatives TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-16 EP disclosed