SCHEMBL7839828

SCHEMBL7839828

CCN(CC)C(=O)C(C1CCNCC1)N1CCC(N)CC1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 8/20 0.38
OPRM1 P35372 7/20 0.38
OPRK1 P41145 2/20 0.38
CPN1 P15169 1/20 0.33
CPB2 Q96IY4 1/20 0.33
GNAI3 P08754 1/20 0.32
GNAO1 P09471 1/20 0.32
GNAI1 P63096 1/20 0.32
MC4R P32245 1/20 0.32
SLC6A2 P23975 3/20 0.32
SLC6A4 P31645 3/20 0.32
SLC6A3 Q01959 3/20 0.32
CACNA2D1 P54289 1/20 0.30
CACNA1B Q00975 1/20 0.30
CACNB1 Q02641 1/20 0.30
SIGMAR1 Q99720 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6586743 0.84 CPN1 (0.32) CPN1CPB2SLC6A2SLC6A4SLC6A3
SCHEMBL6584546 0.82 SLC6A2 (0.35) CPN1CPB2GNAI3GNAO1GNAI1
Hydrochloric Acid SCHEMBL5413829 0.81 OPRD1 (0.54) OPRD1OPRM1OPRK1MC4RSIGMAR1
SCHEMBL6585188 0.79 CPN1 (0.34) CPN1CPB2SLC6A2SLC6A4SLC6A3
SCHEMBL6585899 0.77 SLC6A3 (0.43) CPN1CPB2SLC6A2SLC6A4SLC6A3
SCHEMBL6586012 0.77 SMYD3 (0.32) CPN1CPB2SLC6A2SLC6A4SLC6A3
SCHEMBL6587799 0.75 SLC6A2 (0.31) CPN1CPB2GNAI3GNAO1GNAI1
SCHEMBL6584321 0.74
SCHEMBL6584313 0.74 DPP4 (0.37) CPN1CPB2CACNA2D1CACNA1BCACNB1
SCHEMBL6586715 0.73 CA2 (0.38) CACNA2D1CACNA1BCACNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6294555-B1 SEROTONIN HT3 RECEPTOR ANTAGONIST FOR GASTROINTESTINAL DISORDERS DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 2001-09-25 US disclosed
EP-1076055-A1 1- (1-SUBSTITUTED-4-PIPERIDINYL)METHYL]-4-PIPERIDINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, MEDICINAL COMPOSITIONS CONTAINING THE SAME AND INTERMEDIATES OF THESE COMPOUNDS Dainippon Pharmaceutical Co., Ltd. (JP) 2001-02-14 EP disclosed