SCHEMBL78415

SCHEMBL78415

CNC(=O)CCc1ccc(Cl)c(C(C)(C)C)c1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.48
PYGL P06737 1/20 0.47
KMT2A Q03164 2/20 0.45
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
GRIN1 Q05586 4/20 0.42
GRIN2B Q13224 4/20 0.42
RAF1 P04049 2/20 0.41
BRAF P15056 2/20 0.41
TRPV1 Q8NER1 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MEN1 O00255 1/20 0.39
KCNH2 Q12809 1/20 0.39
NR1H2 P55055 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30791548 0.83 PYGL (0.65) PYGLGRIN1GRIN2BTRPV1ALDH1A1
SCHEMBL28190396 0.83 PYGL (0.65) PYGLGRIN1GRIN2BTRPV1ALDH1A1
SCHEMBL78604 0.79 TSHR (0.38) LMNAMAPTRAF1BRAFALDH1A1
SCHEMBL91334 0.79 PYGL (0.49) GAAPYGLKMT2AGRIN1GRIN2B
SCHEMBL7248605 0.78 GAA (0.74) GAAKMT2ALMNAMAPTALDH1A1
SCHEMBL1750889 0.78 PYGL (0.48) PYGLKMT2AGRIN1GRIN2BTRPV1
SCHEMBL1750381 0.77 PYGL (0.47) PYGLKMT2AGRIN1GRIN2BTRPV1
SCHEMBL30729428 0.75 ALDH1A1 (0.48) PYGLKMT2AMAPTGRIN1GRIN2B
SCHEMBL14387746 0.75 HDAC1 (0.53) MAPTALDH1A1
SCHEMBL12993168 0.74 CYP2C19 (0.56) GAATRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed