SCHEMBL78604

SCHEMBL78604

CNC(=O)OCCc1ccc(Cl)c(C(C)(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
LMNA P02545 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
REN P00797 1/20 0.35
YWHAG P61981 1/20 0.35
APP P05067 1/20 0.35
NR1H4 Q96RI1 3/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CYP2D6 P10635 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRNB2 P17787 1/20 0.34
NFKB1 P19838 1/20 0.34
CHRM3 P20309 1/20 0.34
MAPK1 P28482 1/20 0.34
CHRNA7 P36544 1/20 0.34
CHRNA4 P43681 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL91284 0.81 TSHR (0.43) TSHRSMN1; SMN2KDM4EALDH1A1REN
SCHEMBL78415 0.79 GAA (0.48) LMNAALDH1A1MAPTRAF1BRAF
SCHEMBL78606 0.76 IDO1 (0.39) TSHRLMNAALDH1A1MAPK1MAPT
SCHEMBL10885864 0.74 CYP1A2 (0.50) SMN1; SMN2KDM4EALDH1A1CYP2D6
SCHEMBL1751401 0.73 REN (0.43) TSHRSMN1; SMN2KDM4ERENCHRM5
SCHEMBL11650876 0.71 NPC1 (0.53) SMN1; SMN2KDM4EMAPT
SCHEMBL20234272 0.71 CHRM2 (0.43) SMN1; SMN2LMNACHRM2CHRM4CHRM5
SCHEMBL1751233 0.71 REN (0.51) REN
SCHEMBL78610 0.71 LMNA (0.43) SMN1; SMN2LMNAKDM4ERENMAPK1
SCHEMBL4682925 0.70 REN (0.56) REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed