SCHEMBL7841987

SCHEMBL7841987

O=C1CN=C(c2cccnc2)N1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 1/20 0.53
CYP1A2 P05177 4/20 0.47
ALDH1A1 P00352 2/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2A6 P11509 1/20 0.47
CYP11B1 P15538 12/20 0.47
CYP11B2 P19099 12/20 0.47
CYP2C9 P11712 1/20 0.46
TBXAS1 P24557 1/20 0.46
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
TDP2 O95551 2/20 0.44
NPY5R Q15761 1/20 0.44
BTK Q06187 1/20 0.44
CYP19A1 P11511 4/20 0.43
METAP2 P50579 1/20 0.42
SIRT3 Q9NTG7 1/20 0.42
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4795842 0.80 GABRA1 (0.54) NISCHNPY5RLMNAMAPTHPGD
SCHEMBL13635598 0.74 ALPL (0.50) NISCHCYP1A2ALDH1A1CYP3A4CYP2C9
SCHEMBL16796687 0.72 CYP11B1 (0.48) ALDH1A1CYP11B1CYP11B2CYP19A1MAPT
SCHEMBL16661272 0.71 PIK3CD (0.41) CYP1A2ALDH1A1CYP3A4CYP2A6KDM4E
SCHEMBL9855192 0.71 NISCH (0.53) NISCHNPY5RMETAP2MAPTHSD17B10
SCHEMBL17011756 0.70 CYP1A2 (0.48) CYP1A2ALDH1A1CYP3A4CYP2A6CYP11B1
SCHEMBL2427129 0.69 NISCH (1.00) NISCHCYP1A2ALDH1A1CYP3A4CYP2A6
SCHEMBL4789227 0.69 GABRA1 (0.37) SMN1; SMN2
SCHEMBL9855447 0.69 NISCH (0.47) NISCHALDH1A1LMNAMAPTALOX15
SCHEMBL3161806 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839144-B1 PIPERAZINE DERIVATIVES AS THERAPEUTIC AGENTS KNOLL GMBH (DE) 2001-09-19 EP claimed