SCHEMBL7840741

SCHEMBL7840741

CCOC(=O)Oc1cn(C2CC2)c2c(Cl)c(Cl)ncc2c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.34
KCNH2 Q12809 2/20 0.33
ALDH1A1 P00352 3/20 0.32
POLB P06746 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
CUL4A Q13619 1/20 0.32
TOP2A P11388 3/20 0.32
TOP2B Q02880 3/20 0.32
TNF P01375 2/20 0.31
MAP3K5 Q99683 2/20 0.31
LITAF Q99732 1/20 0.31
KMT2A Q03164 3/20 0.30
TSHR P16473 1/20 0.30
MEN1 O00255 1/20 0.30
MAPT P10636 1/20 0.30
HTT P42858 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7503528 0.90 ADRB2 (0.40) ADRB2KCNH2TOP2ATOP2B
SCHEMBL7851893 0.87 CYP3A4 (0.31) CUL4A
SCHEMBL8692136 0.85 ADRB2 (0.47) ADRB2ALDH1A1POLBCHRM2CHRM1
SCHEMBL7851036 0.85 ALDH1A1 (0.37) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL7842470 0.83 ADRB2 (0.34) ADRB2KCNH2ALDH1A1POLBCHRM2
SCHEMBL7841811 0.83 TDP1 (0.37) ALDH1A1POLBCUL4ATNFKMT2A
SCHEMBL7817401 0.80 ADRB2 (0.47) ADRB2KCNH2ALDH1A1POLBCHRM2
SCHEMBL7840720 0.80 TNF (0.33) ALDH1A1POLBCUL4ATNFKMT2A
SCHEMBL7849137 0.78 KDM4E (0.33) ALDH1A1CUL4ARAB9A
SCHEMBL7848826 0.78 TOP2A (0.39) ALDH1A1POLBCUL4ATOP2ATOP2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726270-B1 Derivatives of 1,6-naphthyridone carboxylic acids BAYER AG (DE) 2001-05-23 EP disclosed
EP-0726270-A1 Derivatives of 1,6-naphthyridine carboxylic acids BAYER AG (DE) 1996-08-14 EP disclosed