SCHEMBL7842823

SCHEMBL7842823

Cc1cc(C)cc(Sc2[nH]c(=O)[nH]c(=O)c2C(C)C)c1.Cc1cc(C)cc(Sc2c(C(C)C)c(=O)[nH]c(=O)n2Cc2ccc3ccccc3n2)c1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.34
HTR7 P34969 1/20 0.34
DPP4 P27487 2/20 0.33
CYP3A4 P08684 1/20 0.33
BRD4 O60885 1/20 0.32
PDE10A Q9Y233 1/20 0.32
ALOX5AP P20292 1/20 0.31
FAP Q12884 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6088008 0.93 DPP4 (0.36) HTR1AHTR7DPP4CYP3A4BRD4
SCHEMBL7853690 0.85 PDE10A (0.36) HTR1AHTR7DPP4CYP3A4BRD4
SCHEMBL7852074 0.84 HTT (0.30) ALDH1A1
SCHEMBL7837061 0.82 TPH1 (0.30) ALDH1A1
SCHEMBL7842857 0.80 GRIN1 (0.39) ALDH1A1
SCHEMBL6086514 0.80 PDE10A (0.40) HTR1AHTR7DPP4CYP3A4BRD4
SCHEMBL6086282 0.78 DAO (0.45) KDM4EALDH1A1
SCHEMBL7855251 0.78 NR3C1 (0.31)
SCHEMBL6086685 0.78 HPGD (0.33) KDM4EALDH1A1
SCHEMBL6088087 0.78 GRIN1 (0.45) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100786-A1 ANTIVIRAL PYRIMIDINEDIONE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF Samjin Pharmaceutical Co., Ltd. (KR) 2001-05-23 EP disclosed
WO-2000061564-A1 ANTIVIRAL PYRIMIDINEDIONE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2000-10-19 WO disclosed