SCHEMBL7842965

SCHEMBL7842965

O=C(NCCc1ccc(OCc2ccccc2)c([N+](=O)[O-])c1)C(F)(F)F

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
CTSV O60911 4/20 0.52
CTSL P07711 4/20 0.52
POLB P06746 3/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
LMNA P02545 1/20 0.50
HTT P42858 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
MAPT P10636 2/20 0.49
PDCD1 Q15116 2/20 0.44
CD274 Q9NZQ7 2/20 0.44
HTR1A P08908 1/20 0.44
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7281747 0.85 MTNR1A (0.55) ALDH1A1MEN1KMT2APOLBLMNA
SCHEMBL29989715 0.83 NPC1 (0.57) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL5913295 0.83 NPC1 (0.57) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL98541 0.80 SMN1; SMN2 (0.43) ALDH1A1KMT2ANPC1RAB9ALMNA
SCHEMBL7840693 0.80 KDM4E (0.57) ALDH1A1MEN1KMT2ACTSVCTSL
SCHEMBL27038529 0.79 POLB (0.54) ALDH1A1MEN1KMT2ACTSVCTSL
SCHEMBL5642071 0.79 CTSV (0.56) ALDH1A1MEN1KMT2ACTSVCTSL
Bromide SCHEMBL11670771 0.79 KDM4E (0.56) ALDH1A1MEN1KMT2ACTSVCTSL
Hydrochloric Acid SCHEMBL11669913 0.79 KDM4E (0.56) ALDH1A1MEN1KMT2ACTSVCTSL
SCHEMBL7339301 0.78 ALDH1A1 (0.46) ALDH1A1POLBNPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0558677-B1 BIOLOGICALLY ACTIVE AMINES ASTRAZENECA AB (SE) 2001-08-16 EP disclosed
US-5763465-A 7-(2-aminoethyl) benzothiazolones ASTRA PHARMACEUTICALS LIMITED (GB) 1998-06-09 US disclosed
US-5648370-A 7-(2-aminoethyl) benzothiazolones ASTRA PHARMACEUTICALS LIMITED (GB) 1997-07-15 US disclosed