SCHEMBL7843584

SCHEMBL7843584

O=C1c2ccccc2CN(CCCO)c2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
SIRT1 Q96EB6 1/20 0.44
DRD2 P14416 3/20 0.41
DRD5 P21918 3/20 0.41
DRD3 P35462 3/20 0.41
HTR1A P08908 1/20 0.41
HTR7 P34969 2/20 0.41
MAOA P21397 1/20 0.41
NPC1 O15118 2/20 0.40
ALDH1A1 P00352 2/20 0.40
RAB9A P51151 2/20 0.40
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
BCHE P06276 1/20 0.39
CES1 P23141 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9375738 0.81 KDM4E (0.65) KDM4EALOX15TSHRSIRT1DRD2
SCHEMBL7839080 0.79 CYP2D6 (0.45) KDM4EALOX15TSHRSIRT1DRD2
SCHEMBL24437908 0.77 KDM4E (0.63) KDM4EALOX15TSHRSIRT1DRD2
SCHEMBL11458214 0.76 NR3C1 (0.53) KDM4EALOX15TSHRSIRT1DRD3
SCHEMBL8013456 0.75 CYP2D6 (0.64) KDM4EALOX15TSHRSIRT1DRD2
SCHEMBL7609349 0.73 SLC6A1 (0.54)
Hydrochloric Acid SCHEMBL7842784 0.73 SLC6A1 (0.53)
SCHEMBL86299 0.73 MAOA (0.50) MAOAALDH1A1MAPTBCHECES1
SCHEMBL91647 0.72 ALDH1A1 (0.42) DRD2DRD5DRD3ALDH1A1CES1
SCHEMBL9466888 0.71 KDM4E (0.69) KDM4EALOX15TSHRSIRT1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820450-B1 N-substituted azaheterocyclic carboxylic acids and alkylesters thereof NOVO NORDISK AS (DK) 2001-09-12 EP disclosed
EP-0820450-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1998-01-28 EP disclosed
WO-1996031497-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1996-10-10 WO disclosed