SCHEMBL7843862

SCHEMBL7843862

CSc1ccc(C(Br)C(=O)c2ccc(F)cc2F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.46
CES1 P23141 3/20 0.46
AKR1C3 P42330 4/20 0.35
AKR1C2 P52895 4/20 0.35
AGBL2 Q5U5Z8 1/20 0.34
PTGS1 P23219 2/20 0.34
PPARG P37231 2/20 0.34
EGFR P00533 1/20 0.34
CYP1A2 P05177 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
MAPT P10636 1/20 0.34
DRD1 P21728 1/20 0.34
MAPK1 P28482 1/20 0.34
PTGS2 P35354 1/20 0.34
OPRM1 P35372 1/20 0.34
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7088208 0.84 CES2 (0.57) CES2CES1AKR1C3AKR1C2AGBL2
SCHEMBL7843292 0.83 CES2 (0.43) CES2CES1AKR1C3AKR1C2MAPT
SCHEMBL7089429 0.80 PLK1 (0.41) CES2CES1AKR1C3AKR1C2MAPT
SCHEMBL7508723 0.80 PLK1 (0.41) CES2CES1AKR1C3AKR1C2MAPT
SCHEMBL7847640 0.78 CES2 (0.49) CES2CES1AKR1C3AKR1C2ALDH1A1
SCHEMBL7814039 0.75 CES2 (0.50) CES2CES1CYP1A2
SCHEMBL6518724 0.74 CES2 (0.57) CES2CES1ALDH1A1L3MBTL1
SCHEMBL7088183 0.74 CES2 (0.62) CES2CES1
SCHEMBL14829993 0.73 CES2 (0.61) CES2CES1ALDH1A1L3MBTL1
SCHEMBL7843732 0.72 KMT2A (0.39) CES2CES1AKR1C3AKR1C2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1125932-A2 Substituted thiazoles for the treatment of inflammation G.D. SEARLE & CO. (US) 2001-08-22 EP disclosed
US-5668161-A Substituted thiazoles for the treatment of inflammation G.D. SEARLE & CO. (US) 1997-09-16 US disclosed