SCHEMBL7847640

SCHEMBL7847640

CSc1ccc(C(Br)C(=O)c2cccc(F)c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.49
CES1 P23141 2/20 0.49
CHRNB2 P17787 1/20 0.43
SLC6A2 P23975 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA4 P43681 1/20 0.43
SLC6A3 Q01959 1/20 0.43
PARP1 P09874 1/20 0.41
ALDH1A1 P00352 5/20 0.40
ESR1 P03372 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
LMNA P02545 2/20 0.38
GAA P10253 2/20 0.38
KDM4E B2RXH2 1/20 0.36
AKR1C3 P42330 2/20 0.36
AKR1C2 P52895 2/20 0.36
PLA2G7 Q13093 1/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7089429 0.82 PLK1 (0.41) CES2CES1ALDH1A1LMNAAKR1C3
SCHEMBL7508723 0.82 PLK1 (0.41) CES2CES1ALDH1A1LMNAAKR1C3
SCHEMBL7845030 0.82 AKR1C3 (0.46) CES2CES1ALDH1A1LMNAKDM4E
SCHEMBL8549601 0.82 CES2 (0.61) CES2CES1CHRNB2SLC6A2CHRNB4
SCHEMBL7843862 0.78 CES2 (0.46) CES2CES1ALDH1A1AKR1C3AKR1C2
Bromide SCHEMBL6285189 0.77 CES2 (0.51) CES2CES1CHRNB2SLC6A2CHRNB4
SCHEMBL7215388 0.77 CA2 (0.54) CES2CES1CHRNB2SLC6A2CHRNB4
SCHEMBL10889643 0.76 CES2 (0.48) CES2CES1ALDH1A1LMNAKDM4E
SCHEMBL7810937 0.76 CES2 (0.52) CES2CES1PARP1ALDH1A1ESR1
SCHEMBL7843096 0.75 PLK1 (0.42) CES2CES1ALDH1A1HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1125932-A2 Substituted thiazoles for the treatment of inflammation G.D. SEARLE & CO. (US) 2001-08-22 EP disclosed
US-5668161-A Substituted thiazoles for the treatment of inflammation G.D. SEARLE & CO. (US) 1997-09-16 US disclosed