SCHEMBL7843940

SCHEMBL7843940

NC(Cc1c[nH]c2cc(Br)ccc12)OC(=O)/C=C/C(=O)OC(N)Cc1c[nH]c2cc(Br)ccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.43
CHRNA7 P36544 1/20 0.43
CHRNA4 P43681 1/20 0.43
BLM P54132 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
PTPRA P18433 1/20 0.42
CYP2A6 P11509 1/20 0.42
SCN9A Q15858 1/20 0.41
CYP2C19 P33261 1/20 0.41
KDM4E B2RXH2 2/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
TSHR P16473 2/20 0.40
PMP22 Q01453 2/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
MPO P05164 1/20 0.40
HIF1A Q16665 1/20 0.40
ADRB3 P13945 1/20 0.40
ITGB2 P05107 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7846486 0.85 GPR84 (0.50) BLMNPSR1PTPRASCN9ACYP2C19
SCHEMBL7997830 0.79 HTR2A (0.53) BLMNPSR1CYP2C19LMNATSHR
SCHEMBL30381776 0.78 KMT2A (0.66) CHRNB2CHRNA7CHRNA4BLMNPSR1
SCHEMBL274624 0.78 KMT2A (0.66) CHRNB2CHRNA7CHRNA4BLMNPSR1
SCHEMBL29855626 0.78 KMT2A (0.66) CHRNB2CHRNA7CHRNA4BLMNPSR1
SCHEMBL8502601 0.78 KMT2A (0.66) CHRNB2CHRNA7CHRNA4BLMNPSR1
SCHEMBL274625 0.78 KMT2A (0.66) CHRNB2CHRNA7CHRNA4BLMNPSR1
SCHEMBL8525797 0.78 TACR1 (0.51) CHRNB2CHRNA7CHRNA4BLMNPSR1
SCHEMBL16976220 0.77 PTPRA (0.51) CHRNB2CHRNA7CHRNA4BLMNPSR1
SCHEMBL19846983 0.77 PTPRA (0.51) CHRNB2CHRNA7CHRNA4BLMNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109784-A1 INDOLINE DERIVATIVES AS 5-HT2B AND/OR 5-HT2C RECEPTOR LIGANDS VERNALIS RESEARCH LIMITED (GB) 2001-06-27 EP disclosed
WO-2000012475-A1 INDOLINE DERIVATIVES AS 5-HT2B AND/OR 5-HT2C RECEPTOR LIGANDS VERNALIS RESEARCH LIMITED (GB) 2000-03-09 WO disclosed