SCHEMBL7844138

SCHEMBL7844138

Cc1[nH]c2ccccc2c1CCBr

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.69
ALDH1A1 P00352 3/20 0.69
TSHR P16473 1/20 0.69
KDM4E B2RXH2 3/20 0.67
POLB P06746 1/20 0.67
HTR6 P50406 1/20 0.65
MAPT P10636 5/20 0.61
CYP3A4 P08684 1/20 0.61
GAA P10253 2/20 0.56
CASP1 P29466 1/20 0.56
CASP7 P55210 1/20 0.56
PABPC1 P11940 1/20 0.52
ALOX15 P16050 1/20 0.52
AHR P35869 1/20 0.52
LMNA P02545 2/20 0.50
KRAS P01116 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
GFER P55789 1/20 0.48
TDP1 Q9NUW8 1/20 0.47
KMT2A Q03164 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11227976 0.91 KDM4E (0.70) HTTALDH1A1TSHRKDM4EPOLB
SCHEMBL8552151 0.83 ALDH1A1 (0.71) HTTALDH1A1TSHRKDM4EPOLB
SCHEMBL28138965 0.83 ALDH1A1 (0.71) HTTALDH1A1TSHRKDM4EPOLB
SCHEMBL29415611 0.81 ALDH1A1 (0.69) HTTALDH1A1TSHRKDM4EPOLB
SCHEMBL9780083 0.81 HTT (0.69) HTTALDH1A1TSHRKDM4EPOLB
SCHEMBL7844388 0.81 ALDH1A1 (1.00) HTTALDH1A1TSHRKDM4EPOLB
SCHEMBL1424220 0.81 ALDH1A1 (0.69) HTTALDH1A1TSHRKDM4EPOLB
SCHEMBL8998008 0.81 KDM4E (0.72) HTTALDH1A1TSHRKDM4EPOLB
SCHEMBL18383120 0.80 MAPT (0.69) HTTALDH1A1TSHRKDM4EPOLB
Hydrochloric Acid SCHEMBL273338 0.80 ALDH1A1 (0.67) HTTALDH1A1TSHRKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106674079-A Synthesis method of panobinostat 南京卡文迪许生物工程技术有限公司 2017-05-17 CN claimed
CN-106674080-A Synthesis method of panobinostat 南京卡文迪许生物工程技术有限公司 2017-05-17 CN claimed
CN-106674080-A Synthesis method of panobinostat 南京卡文迪许生物工程技术有限公司 2017-05-17 CN disclosed
CN-106674079-A Synthesis method of panobinostat 南京卡文迪许生物工程技术有限公司 2017-05-17 CN disclosed
EP-0831824-A4 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2001-05-02 EP disclosed
EP-0831824-A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1998-04-01 EP disclosed
WO-1996039140-A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1996-12-12 WO disclosed
EP-0061333-B1 9-(2-(3-INDOLYL)ETHYL)-1-OXA-4,9-DIAZASPIRO(5.5)UNDECAN-3-ONES SYNTEX (U.S.A.) INC. (US) 1986-01-02 EP disclosed
EP-0061333-A1 9-(2-(3-Indolyl)ethyl)-1-oxa-4,9-diazaspiro(5.5)undecan-3-ones SYNTEX (U.S.A.) INC. (US) 1982-09-29 EP disclosed
US-4332804-A TREATMENT OF HYPERTENSION, CONGESTIVE HEART FAILURE, ARRHYTHMIA, MIGRAINE, VASOSPASTIC DISORDERS AND ASTHMA SYNTEX (U.S.A.) INC. (US) 1982-06-01 US disclosed
US-4110459-A ANALGESIC AMERICAN HOECHST CORPORATION (US) 1978-08-29 US disclosed
US-4101663-A ANTIHYPERTENSIVES AMERICAN HOECHST CORPORATION (US) 1978-07-18 US disclosed
US-4046900-A TRANQUILIZERS, HYPOTENSIVES, ANALGESICS AMERICAN HOECHST CORPORATION (US) 1977-09-06 US disclosed