SCHEMBL7844388

SCHEMBL7844388

Cc1[nH]c2ccccc2c1CCO

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 1.00
HTT P42858 3/20 1.00
TSHR P16473 1/20 1.00
KDM4E B2RXH2 2/20 0.83
POLB P06746 1/20 0.83
HTR6 P50406 1/20 0.65
MAPT P10636 4/20 0.61
CYP3A4 P08684 1/20 0.61
GAA P10253 1/20 0.60
CASP1 P29466 1/20 0.60
CASP7 P55210 1/20 0.60
PABPC1 P11940 1/20 0.56
ALOX15 P16050 1/20 0.56
AHR P35869 1/20 0.52
LMNA P02545 3/20 0.50
KRAS P01116 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7436988 0.91 KDM4E (1.00) ALDH1A1HTTTSHRKDM4EPOLB
SCHEMBL3196770 0.85 ALDH1A1 (0.73) ALDH1A1HTTTSHRKDM4EPOLB
SCHEMBL8552151 0.83 ALDH1A1 (0.71) ALDH1A1HTTTSHRKDM4EPOLB
SCHEMBL28138965 0.83 ALDH1A1 (0.71) ALDH1A1HTTTSHRKDM4EPOLB
SCHEMBL9780083 0.81 HTT (0.69) ALDH1A1HTTTSHRKDM4EPOLB
SCHEMBL29415611 0.81 ALDH1A1 (0.69) ALDH1A1HTTTSHRKDM4EPOLB
SCHEMBL1424220 0.81 ALDH1A1 (0.69) ALDH1A1HTTTSHRKDM4EPOLB
SCHEMBL7844138 0.81 HTT (0.69) ALDH1A1HTTTSHRKDM4EPOLB
SCHEMBL8998008 0.81 KDM4E (0.72) ALDH1A1HTTTSHRKDM4EPOLB
SCHEMBL27824370 0.81 ALDH1A1 (0.68) ALDH1A1HTTTSHRKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115772183-A Indolylethyl fluoroboric acid derivatives, and preparation method and application thereof 复旦大学 2023-03-10 CN disclosed
CN-112430206-B Preparation method of chiral/racemic 6-substituted indole compound 上海交通大学 2022-03-18 CN disclosed
CN-112430206-A Preparation method of chiral/racemic 6-substituted indole compound 上海交通大学 2021-03-02 CN disclosed
US-7745641-B2 Nitrogen-containing heterocyclic compound KYOWA HAKKO KIRIN CO., LTD. (JP) 2010-06-29 US disclosed
EP-2108642-A1 JAK INHIBITOR Kyowa Hakko Kirin Co., Ltd. (JP) 2009-10-14 EP disclosed
US-20090054407-A1 Nitrogen-containing heterocyclic compound KYOWA HAKKO KOGYO CO., LTD. (JP) 2009-02-26 US disclosed
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed
EP-0831824-A4 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2001-05-02 EP disclosed
EP-0831824-A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1998-04-01 EP disclosed
WO-1996039140-A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1996-12-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090054407-A1 Nitrogen-containing heterocyclic compound NR4A1, NR5A2, PRMT8 ALDH1A1 3131/4885HTT 1717/4885TSHR 563/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.