SCHEMBL7845308

SCHEMBL7845308

O=C(C=Cc1cccnc1)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1C(O)C(=O)NC1CCCCC1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
C3AR1 Q16581 8/20 0.50
ALDH1A1 P00352 1/20 0.42
KDM4E B2RXH2 1/20 0.42
CHRNB2 P17787 1/20 0.41
CHRNA7 P36544 1/20 0.41
CHRNA4 P43681 1/20 0.41
ACE P12821 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
FKBP1A P62942 1/20 0.39
NAMPT P43490 2/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7846923 0.86 ACE (0.51) C3AR1ALDH1A1KDM4EACE
SCHEMBL7844050 0.83 ALDH1A1 (0.54) ALDH1A1KDM4EACEMEN1KMT2A
SCHEMBL7853401 0.83 C3AR1 (0.60) C3AR1ALDH1A1KDM4EFKBP1ANAMPT
SCHEMBL7855242 0.80 KDM4E (0.63) ALDH1A1KDM4EACEMEN1KMT2A
SCHEMBL7851592 0.80 ALDH1A1 (0.54) ALDH1A1KDM4EACE
SCHEMBL7853586 0.79 ALDH1A1 (0.49) ALDH1A1KDM4EMEN1KMT2ATDP1
SCHEMBL7844048 0.77 KMT2A (0.45) ALDH1A1KDM4EMEN1KMT2ATDP1
SCHEMBL7855475 0.77 ACE (0.54) ALDH1A1KDM4EACE
SCHEMBL7851487 0.77 SIGMAR1 (0.48) ALDH1A1KDM4ETDP1CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL7851195 0.76 ACE (0.53) ALDH1A1KDM4EACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709373-B1 PYRROLIDINE DERIVATIVE ZAIDAN HOJIN BISEIBUTSU (JP) 2001-10-17 EP disclosed
US-5965556-A KETO-ACID AMIDE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND METHODS FOR INHIBITING THE ACTIVITY OF SERINE PROTEASE OR THIOL PROTEASE BY ADMINISTERING THE DERIVATIVE TO A MAMMAL; ALZHEIMER'S DISEASE ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYUKAI (JP) 1999-10-12 US disclosed
US-5756763-A ENZYME INHIBITOR ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYUKAI (JP) 1998-05-26 US disclosed
EP-0709373-A1 NOVEL PYRROLIDINE DERIVATIVE ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1996-05-01 EP disclosed