SCHEMBL7845370

SCHEMBL7845370

O=C1NCCC(=O)c2c(Br)c[nH]c21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 6/20 0.55
CDK5R1 Q15078 6/20 0.55
CCNB2 O95067 5/20 0.55
CDK1 P06493 5/20 0.55
CCNB1 P14635 5/20 0.55
CCNB3 Q8WWL7 5/20 0.55
CDK4 P11802 3/20 0.55
ERBB2 P04626 2/20 0.55
MAP2K1 Q02750 5/20 0.49
RAF1 P04049 4/20 0.49
MAPK1 P28482 4/20 0.49
PARP10 Q53GL7 3/20 0.39
PARP11 Q9NR21 2/20 0.39
PARP1 P09874 2/20 0.35
HTT P42858 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5558439 0.70 CDK5 (0.41) CDK5CDK5R1CCNB2CDK1CCNB1
SCHEMBL3424550 0.70 CDK5 (0.55) CDK5CDK5R1CCNB2CDK1CCNB1
SCHEMBL1250325 0.70 CDK5 (0.73) CDK5CDK5R1CCNB2CDK1CCNB1
SCHEMBL1250329 0.70 CDK5 (0.73) CDK5CDK5R1CCNB2CDK1CCNB1
SCHEMBL6652262 0.67 MAP2K1 (0.44) CDK5CDK5R1CCNB2CDK1CCNB1
SCHEMBL7837428 0.66 MAP2K1 (1.00) CDK5CDK5R1CCNB2CDK1CCNB1
Aldisin SCHEMBL7844916 0.65 MAP2K1 (1.00) CDK5CDK5R1CCNB2CDK1CCNB1
SCHEMBL3001277 0.65 MAPT (0.52) CDK5CDK5R1CCNB2CDK1CCNB1
SCHEMBL116223 0.65
SCHEMBL3427648 0.63 TUBB4A (0.68) MAP2K1RAF1MAPK1PARP1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711773-B1 HYMENIALDISINE AND DERIVATIVE THEREOF, PROCESS FOR PRODUCING INTERMEDIATE FOR SYNTHESIZING THE SAME, AND SAID INTERMEDIATE SUNTORY LTD (JP) 2001-09-12 EP disclosed
US-5621099-A CARDIOVASCULAR DISORDERS SUNTORY LIMITED (JP) 1997-04-15 US disclosed
EP-0711773-A1 HYMENIALDISINE AND DERIVATIVE THEREOF, PROCESS FOR PRODUCING INTERMEDIATE FOR SYNTHESIZING THE SAME, AND SAID INTERMEDIATE SUNTORY LIMITED (JP) 1996-05-15 EP disclosed