SCHEMBL7846535

SCHEMBL7846535

O=C1C(c2ccc(Cl)c(Cl)c2)CCCN1Cc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 3/20 0.43
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 2/20 0.43
SLC6A3 Q01959 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 1/20 0.42
KCNA5 P22460 1/20 0.42
HTR2C P28335 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24200353 0.85 CHRM2 (0.52) L3MBTL1ALDH1A1
SCHEMBL17138501 0.85 CHRM2 (0.52) L3MBTL1ALDH1A1
SCHEMBL6579768 0.82 PER2 (0.51) SIGMAR1L3MBTL1
SCHEMBL7805639 0.82 PER2 (0.51) SIGMAR1L3MBTL1
SCHEMBL6581110 0.82 PER2 (0.51) SIGMAR1L3MBTL1
SCHEMBL20908736 0.78 POLB (0.50) SIGMAR1
SCHEMBL11258609 0.78 DRD2 (0.53) L3MBTL1
SCHEMBL11382882 0.75 PDE4A (0.49) SIGMAR1ALDH1A1
SCHEMBL2311013 0.74 HTR2C (0.46) OPRK1OPRM1OPRD1SLC6A2SLC6A4
SCHEMBL1280166 0.73 SIGMAR1 (0.43) SIGMAR1SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003743-A4 3,3-DISUBSTITUTED PIPERIDINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO INC (US) 2001-04-11 EP disclosed
EP-1003743-A1 3,3-DISUBSTITUTED PIPERIDINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Merck & Co., Inc. (US) 2000-05-31 EP disclosed
WO-1998031364-A1 3,3-DISUBSTITUTED PIPERIDINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 1998-07-23 WO disclosed