SCHEMBL7846754

SCHEMBL7846754

NC1CON(Cc2ccccc2)C1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
EHMT2 Q96KQ7 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
TSHR P16473 1/20 0.41
AADAT Q8N5Z0 4/20 0.40
F2 P00734 1/20 0.40
PLG P00747 1/20 0.40
ELANE P08246 1/20 0.40
CTSG P08311 1/20 0.40
CMA1 P23946 1/20 0.40
CTRC Q99895 1/20 0.40
EP300 Q09472 1/20 0.39
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38
MGLL Q99685 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18740588 0.84 KMT2A (0.41) ALDH1A1KMT2AMEN1SMN1; SMN2GAA
SCHEMBL18740497 0.84 ALDH1A1 (0.41) ALDH1A1KMT2AMEN1F2CYP1A2
SCHEMBL18740496 0.84 ALDH1A1 (0.41) ALDH1A1KMT2AMEN1F2CYP1A2
SCHEMBL18740587 0.84 KMT2A (0.41) ALDH1A1KMT2AMEN1SMN1; SMN2GAA
Hydrochloric Acid SCHEMBL18740595 0.83 ALDH1A1 (0.41) ALDH1A1KMT2AF2DRD2
Hydrochloric Acid SCHEMBL18740594 0.83 ALDH1A1 (0.41) ALDH1A1KMT2AF2DRD2
SCHEMBL2687303 0.82 HTT (0.46) ALDH1A1KMT2AMEN1GAA
SCHEMBL9566068 0.74 KMT2A (0.42) KMT2AMEN1SMN1; SMN2DRD2DRD4
SCHEMBL2010924 0.71
SCHEMBL11036458 0.70 MEN1 (0.38) ALDH1A1KMT2AMEN1AADATCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0535645-B1 Carbamate derivatives of 4-amino-3-isoxazolidinones and 3-amino-1-hydroxypyrrolidin-2-ones, a process for their preparation and their use as medicaments AVENTIS PHARMA INC (US) 2001-05-09 EP disclosed
EP-1069125-A2 Carbamate derivatives of 4-amino-3-isoxazolidinones, 3-amino-1-hydroxypyrrolidin-2-ones and 1-amino-1-cyclopropanecarboxylic acid analogs, a process for their preparation and their use as medicaments AVENTIS PHARMACEUTICALS INC. (US) 2001-01-17 EP disclosed
US-5234941-A Cognition activators; Alzheimer's disease; cholinergic agents; acetylchloinesterase inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-08-10 US disclosed
US-5231093-A Carbamate derivatives of 4-amino-3-isoxazolidinones, 3-amino-1-hydroxypyrrolidin-2-ones and 1-amino-1-cyclopropanecarboxylic acid analogs HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-27 US disclosed
EP-0535645-A2 Carbamate derivatives of 4-amino-3-isoxazolidinones, 3-amino-1-hydroxypyrrolidin-2-ones and 1-amino-1-cyclopropanecarboxylic acid analogs, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-04-07 EP disclosed
US-5153193-A Nootropic, cholinergic agents HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-10-06 US disclosed
US-4826527-A Aminophenylmethyl isoxazolidinones as plant regulators FMC CORPORATION (US) 1989-05-02 US disclosed