SCHEMBL7848201

SCHEMBL7848201

CCOC(=O)N1CCC2(CC1)NC(=O)N(NC(=O)[C@H](CC(C)C)[C@H](CCCc1ccccc1)C(=O)NOCc1ccccc1)C2=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.36
MMP1 P03956 1/20 0.35
MMP13 P45452 1/20 0.35
ALDH1A1 P00352 5/20 0.35
CYP1A2 P05177 1/20 0.35
POLB P06746 1/20 0.35
CYP2C9 P11712 1/20 0.35
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
TSHR P16473 1/20 0.34
MMP3 P08254 2/20 0.34
HTT P42858 1/20 0.34
CTSL P07711 2/20 0.33
CTSK P43235 2/20 0.33
CTSS P25774 1/20 0.33
LMNA P02545 1/20 0.33
BACE1 P56817 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7955667 0.91 MMP1 (0.40) L3MBTL1MMP1MMP13ALDH1A1CYP1A2
SCHEMBL7957224 0.90 MMP1 (0.38) L3MBTL1MMP1MMP13MMP3CTSL
SCHEMBL7960477 0.90 MMP1 (0.38) L3MBTL1MMP1MMP13MMP3CTSL
SCHEMBL7960470 0.90 MMP1 (0.38) L3MBTL1MMP1MMP13MMP3CTSL
SCHEMBL7957364 0.89 MMP1 (0.39) L3MBTL1MMP1MMP13MMP3CTSL
SCHEMBL7827988 0.89 MMP1 (0.39) L3MBTL1MMP1MMP13MMP3CTSL
SCHEMBL7849143 0.89 HDAC1 (0.41) MMP1MMP13CTSLCTSKCTSS
SCHEMBL7848203 0.88 L3MBTL1 (0.35) L3MBTL1ALDH1A1CYP1A2POLBCYP2C9
SCHEMBL7946779 0.87 MMP1 (0.36) MMP1MMP13POLBMMP3CTSL
SCHEMBL7946782 0.87 MMP1 (0.36) MMP1MMP13POLBMMP3CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1137640-A1 CYCLIC HYDRAZINE DERIVATIVES AS TNF-ALPHA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2001-10-04 EP disclosed
US-6281363-B1 ANTIINFLAMMATORY AGENTS; ANTIARTHRITIC AGENTS; AUTOIMMUNE DISORDERS HOFFMANN-LA ROCHE INC. 2001-08-28 US disclosed
WO-2000035885-A1 CYCLIC HYDRAZINE DERIVATIVES AS TNF-ALPHA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-22 WO disclosed