SCHEMBL7848658

SCHEMBL7848658

CN(C)c1ccc(N(CCc2ccc([N+](=O)[O-])cc2)C(N)=O)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC25C P30307 4/20 0.55
TDP1 Q9NUW8 2/20 0.48
TSHR P16473 2/20 0.48
MAPT P10636 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
MAPK1 P28482 1/20 0.48
PHLPP2 Q6ZVD8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
MEN1 O00255 1/20 0.47
THRB P10828 1/20 0.47
APEX1 P27695 1/20 0.47
RECQL P46063 1/20 0.47
BLM P54132 1/20 0.47
KMT2A Q03164 1/20 0.47
KCNH2 Q12809 5/20 0.46
SIGMAR1 Q99720 1/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29668140 0.87 ALDH1A1 (0.53) CDC25CTDP1TSHRMAPTCYP1A2
SCHEMBL27531317 0.86 CRHBP (0.50) TSHRMAPTCYP1A2L3MBTL1MEN1
SCHEMBL27470018 0.82 L3MBTL1 (0.54) MAPTL3MBTL1MEN1KMT2AKCNH2
SCHEMBL692306 0.79 ALDH1A1 (0.48) TDP1TSHRMAPTCYP1A2CYP3A4
SCHEMBL27799342 0.76 MMP14 (0.50) TDP1TSHRMAPTL3MBTL1MEN1
SCHEMBL21048770 0.76 CDC25C (0.48) CDC25CTSHRCYP1A2CYP3A4MEN1
SCHEMBL13236074 0.75 MAPT (0.53) CDC25CTDP1TSHRMAPTCYP1A2
SCHEMBL1435066 0.75 CRHBP (0.56) TSHRMAPTCYP1A2CYP3A4L3MBTL1
SCHEMBL1435064 0.75 CRHBP (0.55) TSHRMAPTCYP1A2CYP3A4L3MBTL1
SCHEMBL218018 0.74 MAPT (0.78) TDP1TSHRMAPTCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115719-A2 NOVEL AMIDINE DERIVATIVES, THEIR PREPARATION AND APPLICATION AS MEDICINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2001-07-18 EP disclosed
WO-2000017190-A2 AMIDINE DERIVATIVES, THEIR PREPARATION AND APPLICATION AS MEDICINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2000-03-30 WO disclosed