SCHEMBL7848668

SCHEMBL7848668

NC(=O)CC(NCc1cc2ccccc2o1)c1c[nH]c2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.46
MEN1 O00255 2/20 0.43
MAPT P10636 2/20 0.43
KMT2A Q03164 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
POLB P06746 1/20 0.43
RAB9A P51151 1/20 0.43
TACR1 P25103 7/20 0.41
MGAM O43451 3/20 0.40
GAA P10253 3/20 0.40
SI P14410 3/20 0.40
MGAM2 Q2M2H8 3/20 0.40
MC5R P33032 2/20 0.40
MC1R Q01726 2/20 0.40
PKM P14618 1/20 0.38
CTSK P43235 1/20 0.38
CMA1 P23946 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7847455 0.79 TACR1 (0.43) MAOBMEN1MAPTKMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL27785466 0.78 GABRP (0.47) MEN1MAPTKMT2AMGAMGAA
SCHEMBL7848664 0.78 MC5R (0.61) MEN1MAPTKMT2ASMN1; SMN2NPC1
SCHEMBL27763685 0.74 HTR2A (0.49) MEN1MAPTKMT2AMGAMGAA
SCHEMBL7856881 0.74 TACR1 (0.57) MEN1KMT2APOLBTACR1MGAM
SCHEMBL27763691 0.68 MGAM (0.52) MEN1MAPTKMT2AMGAMGAA
SCHEMBL7846982 0.68 BRS3 (0.60) MEN1MAPTKMT2ASMN1; SMN2NPC1
SCHEMBL7062961 0.68 TACR1 (0.76) MEN1KMT2ATACR1
SCHEMBL7848666 0.68 MAPT (0.53) MEN1MAPTKMT2ASMN1; SMN2NPC1
SCHEMBL27777642 0.68 GPR84 (0.56) MEN1MAPTKMT2AMGAMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140914-A1 NON-PEPTIDE NK1 RECEPTORS ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2001-10-10 EP disclosed
WO-2000037462-A1 NON-PEPTIDE NK1 RECEPTORS ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2000-06-29 WO disclosed