SCHEMBL7848716

SCHEMBL7848716

Cc1ccccc1CN1CCCc2ccc(OCCC3CCN(C(=O)c4ccc(C5=NCCN5)cc4)CC3)cc2C1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.52
KMT2A Q03164 1/20 0.42
CHEK2 O96017 3/20 0.41
F10 P00742 2/20 0.38
HRH3 Q9Y5N1 3/20 0.37
ACHE P22303 3/20 0.37
ACACB O00763 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
BCHE P06276 1/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
FABP6 P51161 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PLA2G1B P04054 1/20 0.34
POLB P06746 1/20 0.34
ATG4B Q9Y4P1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7846418 0.88 MCHR1 (0.64) MCHR1CHEK2F10HRH3ACHE
Hydrochloric Acid SCHEMBL7847176 0.85 KMT2A (0.46) KMT2ACHEK2F10HRH3ACACB
SCHEMBL7850512 0.84 MCHR1 (0.57) MCHR1F10HRH3ACHEACACB
Hydrochloric Acid SCHEMBL7852567 0.84 MCHR1 (0.57) MCHR1F10HRH3ACHEACACB
SCHEMBL7838728 0.80 MCHR1 (0.75) MCHR1CHEK2HRH3ACHEACACB
SCHEMBL7846875 0.79 GPR119 (0.50) CHEK2ACACB
SCHEMBL7838157 0.79 HRH3 (0.44) MCHR1KMT2AF10HRH3ACHE
Hydrochloric Acid SCHEMBL7847077 0.79 ACHE (0.47) MCHR1KMT2AF10HRH3ACHE
SCHEMBL7850981 0.77 CHEK2 (0.47) MCHR1KMT2ACHEK2F10HRH3
SCHEMBL7838252 0.76 GPR119 (0.50) CHEK2HRH3ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1122252-A1 NITROGENOUS FUSED HETEROCYCLE COMPOUNDS, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-08 EP claimed
EP-1122252-A1 NITROGENOUS FUSED HETEROCYCLE COMPOUNDS, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-08 EP disclosed