SCHEMBL7848752

SCHEMBL7848752

O=C(NO)c1ccc(Nc2nccs2)cc1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.57
RAB9A P51151 6/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
HDAC6 Q9UBN7 2/20 0.57
AGER Q15109 1/20 0.57
SMN1; SMN2 Q16637 3/20 0.54
LMNA P02545 2/20 0.54
RECQL P46063 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
ADORA2A P29274 7/20 0.53
SCD O00767 1/20 0.51
CYP2C19 P33261 2/20 0.51
POLB P06746 1/20 0.50
MAPT P10636 2/20 0.49
CYP2C9 P11712 1/20 0.49
HSD17B10 Q99714 1/20 0.49
CYP3A4 P08684 1/20 0.49
KDM4E B2RXH2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1180559 0.84 GAA (0.55) NPC1RAB9AMEN1KMT2AAGER
SCHEMBL4600878 0.81 NPC1 (0.73) NPC1RAB9AMEN1KMT2AAGER
SCHEMBL13783968 0.77 HDAC8 (0.53) ADORA2ACYP2C9
SCHEMBL14881017 0.76 MEN1 (0.54) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL3053636 0.76 SYK (0.54) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL3643755 0.76 RAB9A (0.60) NPC1RAB9AMEN1KMT2ASMN1; SMN2
Bromide SCHEMBL2363119 0.75 SYK (0.53) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL20132429 0.75 HDAC6 (0.51) NPC1RAB9AMEN1KMT2AHDAC6
SCHEMBL11589368 0.74 FFAR2 (0.52) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL4287847 0.74 AGER (0.76) NPC1RAB9AMEN1KMT2AAGER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150565-A1 THIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION bioscience AG (DE) 2001-11-07 EP disclosed
WO-2000045635-A1 THIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2000-08-10 WO disclosed