SCHEMBL7853937

SCHEMBL7853937

COc1ccccc1Oc1c(OCCO)nc(-c2nccc(C(N)=O)n2)nc1C(N)=O

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DHPS P49366 15/20 0.57
EDNRA P25101 5/20 0.56
EDNRB P24530 4/20 0.56
ABCC3 O15438 1/20 0.49
ABCC4 O15439 1/20 0.49
NR1I2 O75469 1/20 0.49
ABCB11 O95342 1/20 0.49
NR1H3 Q13133 1/20 0.49
NR1I3 Q14994 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7851035 0.93 EDNRA (0.48) DHPSEDNRAEDNRB
SCHEMBL4061140 0.91 EDNRA (0.67) DHPSEDNRAEDNRBABCC3ABCC4
SCHEMBL4066782 0.85 DHPS (0.66) DHPSEDNRAEDNRB
SCHEMBL7850706 0.84 EDNRA (0.52) DHPSEDNRAEDNRBABCC3ABCC4
SCHEMBL7700296 0.83 EDNRA (0.57) DHPSEDNRAEDNRBABCC3ABCC4
SCHEMBL4060083 0.82 EDNRA (0.64) DHPSEDNRAEDNRB
SCHEMBL4060942 0.81 DHPS (0.56) DHPSEDNRAEDNRB
SCHEMBL6584032 0.80 DHPS (0.55) DHPSEDNRAEDNRBABCC3ABCC4
SCHEMBL6584269 0.80 DHPS (0.62) DHPSEDNRAEDNRBABCC3ABCC4
SCHEMBL5035324 0.79 DHPS (0.53) DHPSEDNRAEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713875-B1 Sulfonamides HOFFMANN LA ROCHE (CH) 2001-03-21 EP claimed
WO-2001049289-A1 PHARMACEUTICAL AND VETERINARY USES OF ENDOTHELIN ANTAGONISTS TEXAS BIOTECHNOLOGY CORPORATION (US) 2001-07-12 WO disclosed
WO-1996016963-A1 SULFONAMIDES AND THEIR USE AS MEDICAMENTS F. HOFFMANN-LA ROCHE AG (CH) 1996-06-06 WO disclosed
EP-0713875-A1 Sulfonamides F. Hoffmann-La Roche AG (CH) 1996-05-29 EP disclosed