SCHEMBL7855306

SCHEMBL7855306

O=C(NCCN1CCOCC1)C(=O)C1CCCN1C(=O)c1ccc(Cl)cc1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.58
HTR1A P08908 1/20 0.58
MAOA P21397 1/20 0.58
MAOB P27338 1/20 0.58
KCNH2 Q12809 1/20 0.58
CD274 Q9NZQ7 1/20 0.58
EPHX2 P34913 2/20 0.52
SMN1; SMN2 Q16637 4/20 0.51
CNR1 P21554 1/20 0.51
MMP2 P08253 2/20 0.50
MMP9 P14780 2/20 0.50
MMP8 P22894 2/20 0.50
MMP13 P45452 2/20 0.50
KMT2A Q03164 3/20 0.48
TDP1 Q9NUW8 1/20 0.48
MAPT P10636 1/20 0.47
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7852457 0.80 ALDH1A1 (0.56) ALDH1A1HTR1AMAOAMAOBKCNH2
SCHEMBL7844655 0.75 CNR1 (0.48) ALDH1A1SMN1; SMN2CNR1
Moclobemide SCHEMBL3408310 0.75 CD274 (1.00) ALDH1A1HTR1AMAOAMAOBKCNH2
Moclobemide SCHEMBL49708 0.75 CD274 (1.00) ALDH1A1HTR1AMAOAMAOBKCNH2
SCHEMBL7844467 0.75 NPC1 (0.65) ALDH1A1SMN1; SMN2MMP2MMP9MMP8
Moclobemide SCHEMBL11475483 0.74 CD274 (0.97) ALDH1A1HTR1AMAOAMAOBKCNH2
SCHEMBL11440161 0.70 ALDH1A1 (0.71) ALDH1A1HTR1AMAOAMAOBKCNH2
SCHEMBL15126028 0.70 POLB (0.61) ALDH1A1KMT2A
SCHEMBL7854391 0.69 NPC1 (0.47) ALDH1A1SMN1; SMN2KMT2AMAPTLMNA
Hydrochloric Acid SCHEMBL11475540 0.69 ALDH1A1 (0.69) ALDH1A1HTR1AMAOAMAOBKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709373-B1 PYRROLIDINE DERIVATIVE ZAIDAN HOJIN BISEIBUTSU (JP) 2001-10-17 EP disclosed
US-5965556-A KETO-ACID AMIDE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND METHODS FOR INHIBITING THE ACTIVITY OF SERINE PROTEASE OR THIOL PROTEASE BY ADMINISTERING THE DERIVATIVE TO A MAMMAL; ALZHEIMER'S DISEASE ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYUKAI (JP) 1999-10-12 US disclosed
US-5756763-A ENZYME INHIBITOR ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYUKAI (JP) 1998-05-26 US disclosed
EP-0709373-A1 NOVEL PYRROLIDINE DERIVATIVE ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1996-05-01 EP disclosed