SCHEMBL7855837

SCHEMBL7855837

NC(CNc1ccccn1)c1nccc(-c2ccccc2-c2c[nH]cn2)n1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.36
FDPS P14324 1/20 0.36
CDK1 P06493 1/20 0.33
CDK4 P11802 1/20 0.33
CCNB1 P14635 1/20 0.33
CCNA2 P20248 1/20 0.33
CCND1 P24385 1/20 0.33
CDK2 P24941 1/20 0.33
CCNA1 P78396 1/20 0.33
CXCR4 P61073 1/20 0.33
FABP1 P07148 1/20 0.32
FABP6 P51161 1/20 0.32
PCSK9 Q8NBP7 1/20 0.32
CYP1A2 P05177 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7021148 0.79 CYP2D6 (0.46) CYP2D6FDPSCXCR4FABP1FABP6
SCHEMBL5099502 0.77 CDK2 (0.44) CDK1CDK4CCNB1CCNA2CCND1
SCHEMBL7854740 0.72 RAB9A (0.40) CYP2D6FDPSCXCR4MEN1ALDH1A1
SCHEMBL7853925 0.71 PIK3CA (0.41) FDPSMEN1ALDH1A1KMT2A
SCHEMBL7022559 0.70 CYP2D6 (0.36) CYP2D6FDPSCDK1CDK4CCNB1
SCHEMBL7851108 0.68 MEN1 (0.36) CYP2D6FDPSCDK2FABP1FABP6
SCHEMBL3758388 0.66 CYP2D6 (0.66) CYP2D6FDPSCXCR4FABP1FABP6
SCHEMBL14198659 0.65 CYP2D6 (0.56) CYP2D6FDPSCXCR4FABP1FABP6
SCHEMBL1831588 0.65 CYP2D6 (0.56) CYP2D6FDPSCXCR4FABP1FABP6
SCHEMBL7015556 0.61 FABP1 (0.41) CYP2D6FDPSCXCR4FABP1FABP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1087963-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 Chiron Corporation (US) 2001-04-04 EP disclosed
WO-1999065897-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 1999-12-23 WO disclosed