SCHEMBL7021148

SCHEMBL7021148

NC(CNc1ccccn1)c1nccc(-c2ccccc2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.46
AURKA O14965 1/20 0.42
HSP90AA1 P07900 1/20 0.42
PRKACA P17612 1/20 0.42
ADORA2A P29274 1/20 0.42
FDPS P14324 1/20 0.42
FABP1 P07148 1/20 0.41
FABP6 P51161 1/20 0.41
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
F11 P03951 1/20 0.39
CXCR4 P61073 1/20 0.39
HRH4 Q9H3N8 6/20 0.37
GABRA5 P31644 1/20 0.36
PCSK9 Q8NBP7 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.35
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7853925 0.85 PIK3CA (0.41) FDPSMEN1NPC1RAB9AKMT2A
SCHEMBL7854740 0.85 RAB9A (0.40) CYP2D6FDPSMEN1NPC1RAB9A
SCHEMBL7022559 0.82 CYP2D6 (0.36) CYP2D6FDPSFABP1FABP6NPC1
SCHEMBL7855837 0.79 CYP2D6 (0.36) CYP2D6FDPSFABP1FABP6MEN1
SCHEMBL7851108 0.77 MEN1 (0.36) CYP2D6FDPSFABP1FABP6MEN1
SCHEMBL3758388 0.75 CYP2D6 (0.66) CYP2D6FDPSFABP1FABP6CXCR4
SCHEMBL7015556 0.75 FABP1 (0.41) CYP2D6FDPSFABP1FABP6CXCR4
SCHEMBL2331522 0.75 F11 (0.51) CYP2D6AURKAHSP90AA1PRKACAADORA2A
SCHEMBL6644446 0.73 CYP2D6 (0.38) CYP2D6FDPSFABP1FABP6MEN1
SCHEMBL5100516 0.72 VCP (0.47) AURKAHSP90AA1PRKACAADORA2AFABP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317433-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2003-06-11 EP disclosed
WO-2002020495-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2002-03-14 WO disclosed