SCHEMBL78581

SCHEMBL78581

CC(C)(C)c1cc(O)cc(-c2ccccc2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.58
GABRB2 P47870 1/20 0.58
EGFR P00533 2/20 0.57
RXRB P28702 7/20 0.50
RXRA P19793 6/20 0.50
RXRG P48443 3/20 0.50
ABL1 P00519 2/20 0.44
ABCB1 P08183 2/20 0.44
BCR P11274 2/20 0.44
MMP3 P08254 1/20 0.43
BCL2L1 Q07817 1/20 0.43
KIF11 P52732 1/20 0.43
LMNA P02545 1/20 0.41
TYR P14679 1/20 0.41
HSD17B1 P14061 1/20 0.41
HSD17B2 P37059 1/20 0.41
ESR1 P03372 2/20 0.41
ESR2 Q92731 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29771943 0.86 ABL1 (0.60) GABRA1GABRB2EGFRRXRBRXRA
SCHEMBL28857358 0.86 ABL1 (0.60) GABRA1GABRB2EGFRRXRBRXRA
SCHEMBL5546207 0.85 RXRB (0.53) EGFRRXRBRXRARXRGKIF11
SCHEMBL26149393 0.85 RXRB (0.53) EGFRRXRBRXRARXRGKIF11
SCHEMBL11646120 0.85 RXRB (0.59) GABRA1GABRB2EGFRRXRBRXRA
SCHEMBL27757672 0.83 RXRB (0.62) GABRA1GABRB2EGFRRXRBRXRA
SCHEMBL30096028 0.83 RXRB (0.57) GABRA1GABRB2EGFRRXRBRXRA
Phenol SCHEMBL7858678 0.81 GABRA1 (0.73) GABRA1GABRB2EGFRRXRBRXRA
SCHEMBL29561009 0.81 GABRA1 (0.71) GABRA1GABRB2EGFRRXRBRXRA
SCHEMBL25383551 0.80 RXRA (0.59) GABRA1GABRB2RXRBRXRARXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed