SCHEMBL7858451

SCHEMBL7858451

O=C1CN=C(c2ccccc2)c2ccccc2N1CCCC(F)(F)F

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.63
HDAC1 Q13547 1/20 0.63
HDAC8 Q9BY41 1/20 0.63
HDAC6 Q9UBN7 1/20 0.63
NPSR1 Q6W5P4 2/20 0.62
GABRA1 P14867 2/20 0.57
GABRG2 P18507 2/20 0.57
GABRB3 P28472 2/20 0.57
GABRA5 P31644 2/20 0.57
GABRA3 P34903 2/20 0.57
GABRA2 P47869 2/20 0.57
GABRB2 P47870 2/20 0.57
CCKBR P32239 1/20 0.57
GAA P10253 2/20 0.56
HTT P42858 1/20 0.56
GPR55 Q9Y2T6 1/20 0.56
NR1I2 O75469 1/20 0.56
ADORA3 P0DMS8 1/20 0.56
OPRM1 P35372 1/20 0.56
OPRK1 P41145 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3249926 0.85 NR1I2 (0.74) HDAC3HDAC1HDAC8HDAC6NPSR1
SCHEMBL9380657 0.83 HDAC3 (0.69) HDAC3HDAC1HDAC8HDAC6NPSR1
SCHEMBL8851595 0.81 GABRA1 (0.68) HDAC3HDAC1HDAC8HDAC6NPSR1
SCHEMBL1368126 0.80 HDAC3 (0.78) HDAC3HDAC1HDAC8HDAC6NPSR1
SCHEMBL6985755 0.79 GABRA1 (0.65) HDAC3HDAC1HDAC8HDAC6NPSR1
SCHEMBL7541208 0.78 GABRA1 (0.68) HDAC3HDAC1HDAC8HDAC6NPSR1
SCHEMBL27562818 0.77 NPSR1 (0.78) HDAC3HDAC1HDAC8HDAC6NPSR1
SCHEMBL11576361 0.77 GABRA1 (0.62) HDAC3HDAC1HDAC8HDAC6NPSR1
SCHEMBL4414577 0.77 GABRP (0.59) HDAC3HDAC1HDAC8HDAC6GABRA1
SCHEMBL1367380 0.77 HDAC3 (0.98) HDAC3HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1089981-A1 COMPOUNDS FOR INHIBITING BETA-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS. Elan Pharmaceuticals, Inc. (US) 2001-04-11 EP disclosed
WO-1999067220-A1 COMPOUNDS FOR INHIBITING BETA-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS ELAN PHARMACEUTICALS, INC. (US) 1999-12-29 WO disclosed