SCHEMBL7858736

SCHEMBL7858736

COc1ccc(CCOc2cc(SC(CCCCc3ccccc3)CC(=O)NO)ncc2OC)cc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 11/20 0.50
PDE4B Q07343 11/20 0.50
PDE4C Q08493 11/20 0.50
PDE4D Q08499 11/20 0.50
MMP3 P08254 9/20 0.50
MMP1 P03956 8/20 0.50
MMP2 P08253 8/20 0.50
MMP9 P14780 1/20 0.42
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
ALOX5 P09917 1/20 0.40
CSNK2A2 P19784 1/20 0.40
CSNK2A1 P68400 1/20 0.40
EGFR P00533 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6424724 0.82 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DMMP3
SCHEMBL6823664 0.80 MMP3 (0.62) PDE4APDE4BPDE4CPDE4DMMP3
SCHEMBL6819981 0.75 PDE4A (0.62) PDE4APDE4BPDE4CPDE4DMMP3
SCHEMBL6825876 0.72 MMP2 (0.60) PDE4APDE4BPDE4CPDE4DMMP3
SCHEMBL6422449 0.71 PDE4A (0.87) PDE4APDE4BPDE4CPDE4DMMP3
SCHEMBL6822907 0.71 HDAC1 (0.52) PDE4APDE4BPDE4CPDE4DMMP3
SCHEMBL6422312 0.70 PDE4A (0.58) PDE4APDE4BPDE4CPDE4DMMP3
SCHEMBL6823533 0.69 SIRT5 (0.56) PDE4APDE4BPDE4CPDE4DMMP3
SCHEMBL8891569 0.69 KDM4E (0.52) MTNR1AMTNR1BALOX5CSNK2A2CSNK2A1
SCHEMBL6424681 0.68 PDE4A (0.67) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306873-B1 Substituted β-thiocarboxylic acids AVENTIS PHARMACEUTICALS PRODUCTS INC. 2001-10-23 US disclosed