SCHEMBL7858744

SCHEMBL7858744

O=C(O)C(O)(CCN1CCCC1)P(=O)(O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
ARG1 P05089 5/20 0.41
ARG2 P78540 4/20 0.41
CYP2D6 P10635 3/20 0.40
CHRM2 P08172 3/20 0.40
CHRM1 P11229 3/20 0.40
KCNH2 Q12809 3/20 0.40
HTR1A P08908 2/20 0.40
OPRM1 P35372 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
LMNA P02545 1/20 0.40
MAPK1 P28482 2/20 0.39
CYP1A2 P05177 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAPT P10636 3/20 0.38
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL136428 0.77 CA12 (0.47) CA12CA1CA2CA9CYP2D6
SCHEMBL3225341 0.76 CA12 (0.46) CA12CA1CA2CA9CYP2D6
SCHEMBL6222263 0.76 CA12 (0.49) CA12CA1CA2CA9CYP2D6
SCHEMBL9298865 0.76 CA12 (0.49) CA12CA1CA2CA9CYP2D6
SCHEMBL9615006 0.73 FDPS (0.45) CA12CA1CA2CA9CYP2D6
SCHEMBL8630496 0.73 CYP2D6 (0.49) ARG1ARG2CYP2D6CHRM2CHRM1
SCHEMBL18161704 0.73 CA12 (0.40) CA12CA1CA2CA9CYP2D6
SCHEMBL8630883 0.72 CYP2D6 (0.47) ARG1ARG2CYP2D6CHRM2CHRM1
SCHEMBL3067217 0.70 CA12 (0.41) CA12CA1CA2CA9CYP2D6
SCHEMBL27911982 0.69 ARG1 (0.45) ARG1ARG2CYP2D6CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0788362-B1 PHOSPONOCARBOXYLATE COMPOUNDS FOR TREATING ABNORMAL CALCIUM AND PHOSPHATE METABOLISM PROCTER & GAMBLE PHARMA (US) 2001-07-25 EP disclosed
CN-1048017-C Phosphonocarboxylate compounds and pharmaceutical compositions containing the same PROCTER & GAMBLE PHARMA (US) 2000-01-05 CN disclosed
CN-1230409-A Phosphonocarboxylate compounds and pharmaceutical compositions containing the same PROCTER & GAMBLE PHARMA (US) 1999-10-06 CN disclosed
CN-1224018-A Phosphonic carboxylate compounds, pharmaceutical compositions contg. same PROCTER & GAMBLE PHARMA (US) 1999-07-28 CN disclosed
US-5760021-A TREATING OR PREVENTING METABOLIC BONE DISORDERS THE PROCTER & GAMBLE COMPANY (US) 1998-06-02 US disclosed
EP-0788362-A1 PHOSPONOCARBOXYLATE COMPOUNDS FOR TREATING ABNORMAL CALCIUM AND PHOSPHATE METABOLISM PROCTER & GAMBLE PHARMACEUTICALS, INC. (US) 1997-08-13 EP disclosed
CN-1089613-A Phosphonocarboxylate compounds and pharmaceutical compositions containing the same PROCTER & GAMBLE PHARMA (US) 1994-07-20 CN disclosed
WO-1993024131-A1 PHOSPONOCARBOXYLATE COMPOUNDS FOR TREATING ABNORMAL CALCIUM AND PHOSPHATE METABOLISM PROCTER & GAMBLE PHARMACEUTICALS, INC. (US) 1993-12-09 WO disclosed