SCHEMBL7859043

SCHEMBL7859043

Clc1ccc(-c2ccc3c(c2)CNCCO3)cn1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 3/20 0.45
S1PR3 Q99500 2/20 0.45
ASIC3 Q9UHC3 2/20 0.39
PIK3CD O00329 1/20 0.37
CD274 Q9NZQ7 1/20 0.37
DYRK1A Q13627 1/20 0.37
CYP2A6 P11509 1/20 0.36
NPC1 O15118 3/20 0.35
RAB9A P51151 2/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
ACHE P22303 1/20 0.34
NOTUM Q6P988 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3754485 0.84 DYRK1A (0.46) S1PR1S1PR3ASIC3PIK3CDCD274
Hydrochloric Acid SCHEMBL859783 0.78 TGFBR1 (0.42) S1PR1S1PR3ASIC3CD274DYRK1A
SCHEMBL12998010 0.77 PIK3CA (0.54) S1PR1S1PR3ASIC3PIK3CDCYP2A6
SCHEMBL3797512 0.77 S1PR1 (0.45) S1PR1S1PR3ASIC3CD274DYRK1A
SCHEMBL2724081 0.77 ASIC3 (0.37) S1PR1S1PR3ASIC3PIK3CDCD274
SCHEMBL3793368 0.76 HCAR3 (0.39) S1PR1S1PR3ASIC3DYRK1AMAPT
Hydrochloric Acid SCHEMBL3281306 0.76 CD274 (0.43) S1PR1S1PR3ASIC3CD274DYRK1A
SCHEMBL20565297 0.75 PNMT (0.53) S1PR1S1PR3ACHE
SCHEMBL30174754 0.75 PNMT (0.53) S1PR1S1PR3ACHE
Hydrochloric Acid SCHEMBL9278402 0.74 PIK3CD (0.51) S1PR1S1PR3PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118208-A1 BENZOXAZEPIN-4- (5H) -YL DERIVATIVES AND THEIR USE TO TREAT CANCER EXELIXIS, INC. (US) 2010-10-14 WO disclosed