SCHEMBL7859366

SCHEMBL7859366

C=CCOc1ccc(C=O)cc1-c1c(-c2ccc(OC)cc2)noc1-c1ccc(OC)cc1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.41
FLT3 P36888 1/20 0.40
PTGS1 P23219 1/20 0.38
PDE3A Q14432 1/20 0.38
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5729956 0.79 PTGS2 (0.56) PTGS2PTGS1PDE3A
SCHEMBL5730259 0.79 PTGS2 (0.56) PTGS2PTGS1PDE3A
SCHEMBL7846360 0.71 PPARD (0.33) ALDH1A1
SCHEMBL5730289 0.69 MEN1 (0.43) PTGS2PTGS1PDE3A
SCHEMBL5729672 0.69 PTGS2 (0.70) PTGS2PTGS1PDE3A
SCHEMBL3925069 0.69 ALDH1A1 (0.50) ALDH1A1
SCHEMBL29652045 0.68 FDPS (0.71) ALDH1A1
SCHEMBL1396839 0.68 FDPS (0.71) ALDH1A1
SCHEMBL1748511 0.68 ALDH1A1 (0.66) ALDH1A1
SCHEMBL6772444 0.68 TRIM24 (0.47) PTGS2PTGS1PDE3AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102755-A1 SUBSTITUTED ISOXAZOLE DERIVATIVES AS ESTROGEN RECEPTOR MODULATORS CHIRON CORPORATION (US) 2001-05-30 EP disclosed
WO-2000008001-A1 SUBSTITUTED ISOXAZOLE AS ESTROGEN RECEPTOR MODULATORS CHIRON CORPORATION (US) 2000-02-17 WO disclosed