SCHEMBL7861399

SCHEMBL7861399

COc1ccc(COc2ccccc2OC(Cc2ccccc2)C2=NCCN2)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 9/20 0.47
ADRA2B P18089 9/20 0.47
ADRA2C P18825 9/20 0.47
MAOA P21397 10/20 0.47
MAOB P27338 10/20 0.47
NISCH Q9Y2I1 8/20 0.47
ABCB1 P08183 1/20 0.45
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
SGMS2 Q8NHU3 1/20 0.41
AOC3 Q16853 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7854564 1.00 ADRA2A (0.47) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL3169171 0.91 NISCH (0.52) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL9197682 0.89 ADRA2B (0.61) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL9206145 0.89 ADRA2B (0.60) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL7860101 0.87 ADRA2A (0.46) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL7854333 0.87 ADRA2B (0.46) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL7859921 0.87 ADRA2B (0.46) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL9199669 0.85 ADRA2B (0.64) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL9201690 0.83 ADRA2B (0.67) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL7861283 0.83 ADRA2A (0.50) ADRA2AADRA2BADRA2CMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625969-B1 ARYLALKOXYPHENOXY-IMIDAZOLINE COMPOUNDS MERRELL PHARMA INC (US) 2001-03-07 EP disclosed