SCHEMBL7860101

SCHEMBL7860101

Clc1ccc(COc2ccccc2OC(Cc2ccccc2)C2=NCCN2)cc1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 9/20 0.46
ADRA2B P18089 9/20 0.46
ADRA2C P18825 9/20 0.46
MAOA P21397 8/20 0.46
MAOB P27338 8/20 0.46
NISCH Q9Y2I1 7/20 0.46
CCR5 P51681 1/20 0.40
SGMS2 Q8NHU3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3169171 0.93 NISCH (0.52) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL7854333 0.89 ADRA2B (0.46) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL7859921 0.89 ADRA2B (0.46) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL7854564 0.87 ADRA2A (0.47) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL7861399 0.87 ADRA2A (0.47) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL3677271 0.87 NISCH (0.49) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL7861142 0.85 ADRA2A (0.50) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL7861283 0.85 ADRA2A (0.50) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL9204696 0.83 NISCH (0.58) ADRA2AADRA2BADRA2CMAOAMAOB
SCHEMBL9201690 0.83 ADRA2B (0.67) ADRA2AADRA2BADRA2CMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625969-B1 ARYLALKOXYPHENOXY-IMIDAZOLINE COMPOUNDS MERRELL PHARMA INC (US) 2001-03-07 EP disclosed
US-5407954-A Serotonin antagonism; treats depression, anxiety, hypertension and migraine headaches MERRELL DOW PHARMACEUTICALS INC. (US) 1995-04-18 US disclosed
US-5216008-A Antidepressant, anxiolytic, hypotensive and also treats migraine headaches MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-01 US disclosed